BindingDB PrimarySearch

Found 2 hits Enz. Inhib. hit(s) with Target = 'Neuropeptide Y receptor type 1' and Ligand = 'BDBM50296881'
Target/Host (Institution)	Ligand	Target/Host Links	Ligand Links	Trg + Lig Links	Ki nM	ΔG° kJ/mole	IC50 nM	Kd nM	EC50/IC50 nM	k_off s^-1	k_on M^-1s^-1	pH	Temp °C
Neuropeptide Y receptor type 1 (Homo sapiens (Human))	BDBM50296881 ((1-((1R,4R)-4-((S)-2,2-difluoro-1-(4-methoxyphenyl...) Show SMILES Show InChI	PDB Reactome pathway KEGG UniProtKB/SwissProt antibodypedia GoogleScholar AffyNet	CHEMBL PC cid PC sid UniChem Similars	Article PubMed	22	n/a	n/a	n/a	n/a	n/a	n/a	n/a	n/a
Tsukuba Research Institute Curated by ChEMBL					Assay Description Displacement of [125I]PYY from human recombinant neuropeptide Y1 receptor expressed in CHO (NFAT-bla) cells by scintillation counting				Bioorg Med Chem Lett 19: 4781-5 (2009) Article DOI: 10.1016/j.bmcl.2009.06.050 BindingDB Entry DOI: 10.7270/Q2319VXR
Tsukuba Research Institute Curated by ChEMBL					More data for this Ligand-Target Pair
Neuropeptide Y receptor type 1 (Homo sapiens (Human))	BDBM50296881 ((1-((1R,4R)-4-((S)-2,2-difluoro-1-(4-methoxyphenyl...) Show SMILES Show InChI	PDB Reactome pathway KEGG UniProtKB/SwissProt antibodypedia GoogleScholar AffyNet	CHEMBL PC cid PC sid UniChem Similars	Article PubMed	n/a	n/a	280	n/a	n/a	n/a	n/a	n/a	n/a
Tsukuba Research Institute Curated by ChEMBL					Assay Description Antagonist activity at human neuropeptide Y1 receptor expressed in HEK293 cells by [35S]GTPgammaS binding assay				Bioorg Med Chem Lett 19: 4781-5 (2009) Article DOI: 10.1016/j.bmcl.2009.06.050 BindingDB Entry DOI: 10.7270/Q2319VXR
Tsukuba Research Institute Curated by ChEMBL					More data for this Ligand-Target Pair