Target/Host (Institution) | Ligand | Target/Host Links | Ligand Links | Trg + Lig Links | Ki nM | ΔG° kJ/mole | IC50 nM | Kd nM | EC50/IC50 nM | koff s-1 | kon M-1s-1 | pH | Temp °C |
---|---|---|---|---|---|---|---|---|---|---|---|---|---|
PAS domain-containing serine/threonine-protein kinase (Homo sapiens (Human)) | BDBM50154943 (CHEMBL3775576) | PDB MMDB KEGG UniProtKB/SwissProt B.MOAD antibodypedia GoogleScholar AffyNet | CHEMBL PC cid PC sid UniChem Similars | Article PubMed | n/a | n/a | 260 | n/a | n/a | n/a | n/a | n/a | n/a |
Merck KGaA Curated by ChEMBL | Assay Description Inhibition of PASK (unknown origin) | Bioorg Med Chem Lett 26: 1443-51 (2016) Article DOI: 10.1016/j.bmcl.2016.01.062 BindingDB Entry DOI: 10.7270/Q2NZ89G6 | |||||||||||
More data for this Ligand-Target Pair |