Target/Host (Institution) | Ligand | Target/Host Links | Ligand Links | Trg + Lig Links | Ki nM | ΔG° kJ/mole | IC50 nM | Kd nM | EC50/IC50 nM | koff s-1 | kon M-1s-1 | pH | Temp °C |
---|---|---|---|---|---|---|---|---|---|---|---|---|---|
Peroxisome proliferator-activated receptor delta (Homo sapiens (Human)) | BDBM50103947 (3-(4-((5-(4-bromophenyl)-1,2,4-oxadiazol-3-yl)meth...) | PDB UniProtKB/SwissProt antibodypedia GoogleScholar AffyNet | CHEMBL PC cid PC sid UniChem Similars | Article PubMed | n/a | n/a | n/a | n/a | 790 | n/a | n/a | n/a | n/a |
National Institute of Pharmaceutical Education and Research Curated by ChEMBL | Assay Description Agonist activity at human PPARdelta expressed in african green monkey CV1 cells cotransfected with Gal4 assessed as reporter activty by transient tra... | Eur J Med Chem 43: 2784-91 (2008) Article DOI: 10.1016/j.ejmech.2008.01.017 BindingDB Entry DOI: 10.7270/Q2W095QK | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Peroxisome proliferator-activated receptor delta (Homo sapiens (Human)) | BDBM50103947 (3-(4-((5-(4-bromophenyl)-1,2,4-oxadiazol-3-yl)meth...) | PDB UniProtKB/SwissProt antibodypedia GoogleScholar AffyNet | CHEMBL PC cid PC sid UniChem Similars | PubMed | n/a | n/a | n/a | n/a | 790 | n/a | n/a | n/a | n/a |
GlaxoSmithKline Curated by ChEMBL | Assay Description Agonist activity against human PPAR delta receptor in CV-1 cell was determined | Bioorg Med Chem Lett 11: 2385-8 (2001) BindingDB Entry DOI: 10.7270/Q2CJ8CSF | |||||||||||
More data for this Ligand-Target Pair |