Target/Host (Institution) | Ligand | Target/Host Links | Ligand Links | Trg + Lig Links | Ki nM | ΔG° kJ/mole | IC50 nM | Kd nM | EC50/IC50 nM | koff s-1 | kon M-1s-1 | pH | Temp °C |
---|---|---|---|---|---|---|---|---|---|---|---|---|---|
Phosphatidylinositol 4-kinase beta (Homo sapiens (Human)) | BDBM50363167 (CHEMBL1945559) | PDB UniProtKB/SwissProt GoogleScholar AffyNet | CHEMBL PC cid PC sid PDB UniChem | Article PubMed | n/a | n/a | 2.50E+3 | n/a | n/a | n/a | n/a | n/a | n/a |
Ludwig-Maximilians University of Munich Curated by ChEMBL | Assay Description Inhibition of PI4Kbeta using ATP as substrate | J Med Chem 55: 403-13 (2012) Article DOI: 10.1021/jm201286z BindingDB Entry DOI: 10.7270/Q20G3KK7 | |||||||||||
More data for this Ligand-Target Pair |