Target/Host (Institution) | Ligand | Target/Host Links | Ligand Links | Trg + Lig Links | Ki nM | ΔG° kJ/mole | IC50 nM | Kd nM | EC50/IC50 nM | koff s-1 | kon M-1s-1 | pH | Temp °C |
---|---|---|---|---|---|---|---|---|---|---|---|---|---|
Phospholipase A2, major isoenzyme (Sus scrofa (pig)) | BDBM50269843 (Bolinaquinone | CHEMBL477692) | PDB MMDB KEGG UniProtKB/SwissProt B.MOAD DrugBank GoogleScholar AffyNet | CHEMBL PC cid PC sid UniChem Similars | PubMed | n/a | n/a | 400 | n/a | n/a | n/a | n/a | n/a | n/a |
Università degli Studi di Napoli Federico II Curated by ChEMBL | Assay Description Inhibition of pig pancreatic group 1 secretory phospholipase A2 by liquid scintillation counting | J Nat Prod 64: 612-5 (2001) BindingDB Entry DOI: 10.7270/Q28915MQ | |||||||||||
More data for this Ligand-Target Pair |