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Compile Data Set for Download or QSAR

Found 1 hit Enz. Inhib. hit(s) with Target = 'Platelet activating factor receptor' and Ligand = 'BDBM50038764'   
Target/Host
(Institution)
LigandTarget/Host
Links
Ligand
Links
Trg + Lig
Links
Ki
nM
ΔG°
kJ/mole
IC50
nM
Kd
nM
EC50/IC50
nM
koff
s-1
kon
M-1s-1
pHTemp
°C
Platelet activating factor receptor


(Cavia porcellus)
BDBM50038764
PNG
((6-Methoxy-1H-indol-3-yl)-((R)-2-pyridin-3-yl-thia...)
Show SMILES COc1ccc2c(c[nH]c2c1)C(=O)[C@@H]1CSC(N1)c1cccnc1
Show InChI InChI=1S/C18H17N3O2S/c1-23-12-4-5-13-14(9-20-15(13)7-12)17(22)16-10-24-18(21-16)11-3-2-6-19-8-11/h2-9,16,18,20-21H,10H2,1H3/t16-,18?/m0/s1
MMDB

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PC cid
PC sid
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PubMed
9.5n/an/an/an/an/an/an/an/a



Abbott Laboratories

Curated by ChEMBL


Assay Description
Antagonist activity against platelet activating factor (PAF) receptor in rabbit platelet membranes using [3H]C18-PAF as radioligand


J Med Chem 37: 2011-32 (1994)


BindingDB Entry DOI: 10.7270/Q2GH9JM7
More data for this
Ligand-Target Pair