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Compile Data Set for Download or QSAR

Found 1 hit Enz. Inhib. hit(s) with Target = 'Platelet activating factor receptor' and Ligand = 'BDBM50038767'   
Target/Host
(Institution)
LigandTarget/Host
Links
Ligand
Links
Trg + Lig
Links
Ki
nM
ΔG°
kJ/mole
IC50
nM
Kd
nM
EC50/IC50
nM
koff
s-1
kon
M-1s-1
pHTemp
°C
Platelet activating factor receptor


(Cavia porcellus)
BDBM50038767
PNG
((6-Fluoro-1H-indol-3-yl)-((R)-2-pyridin-3-yl-thiaz...)
Show SMILES Fc1ccc2c(c[nH]c2c1)C(=O)[C@@H]1CSC(N1)c1cccnc1
Show InChI InChI=1S/C17H14FN3OS/c18-11-3-4-12-13(8-20-14(12)6-11)16(22)15-9-23-17(21-15)10-2-1-5-19-7-10/h1-8,15,17,20-21H,9H2/t15-,17?/m0/s1
MMDB

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PC cid
PC sid
UniChem
PubMed
5.60n/an/an/an/an/an/an/an/a



Abbott Laboratories

Curated by ChEMBL


Assay Description
Antagonist activity against platelet activating factor (PAF) receptor in rabbit platelet membranes using [3H]C18-PAF as radioligand


J Med Chem 37: 2011-32 (1994)


BindingDB Entry DOI: 10.7270/Q2GH9JM7
More data for this
Ligand-Target Pair