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Compile Data Set for Download or QSAR

Found 1 hit Enz. Inhib. hit(s) with Target = 'Platelet activating factor receptor' and Ligand = 'BDBM50038789'   
Target/Host
(Institution)
LigandTarget/Host
Links
Ligand
Links
Trg + Lig
Links
Ki
nM
ΔG°
kJ/mole
IC50
nM
Kd
nM
EC50/IC50
nM
koff
s-1
kon
M-1s-1
pHTemp
°C
Platelet activating factor receptor


(Cavia porcellus)
BDBM50038789
PNG
(5,6-Dimethoxy-3-((R)-2-pyridin-3-yl-thiazolidine-4...)
Show SMILES COc1cc2c(cn(C(=O)N(C)C)c2cc1OC)C(=O)[C@@H]1CSC(N1)c1cccnc1
Show InChI InChI=1S/C22H24N4O4S/c1-25(2)22(28)26-11-15(14-8-18(29-3)19(30-4)9-17(14)26)20(27)16-12-31-21(24-16)13-6-5-7-23-10-13/h5-11,16,21,24H,12H2,1-4H3/t16-,21?/m0/s1
MMDB

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10n/an/an/an/an/an/an/an/a



Abbott Laboratories

Curated by ChEMBL


Assay Description
Antagonist activity against platelet activating factor (PAF) receptor in rabbit platelet membranes using [3H]C18-PAF as radioligand


J Med Chem 37: 2011-32 (1994)


BindingDB Entry DOI: 10.7270/Q2GH9JM7
More data for this
Ligand-Target Pair