Target/Host (Institution) | Ligand | Target/Host Links | Ligand Links | Trg + Lig Links | Ki nM | ΔG° kJ/mole | IC50 nM | Kd nM | EC50/IC50 nM | koff s-1 | kon M-1s-1 | pH | Temp °C |
---|---|---|---|---|---|---|---|---|---|---|---|---|---|
Platelet glycoprotein 4 (Rattus norvegicus) | BDBM263256 (US9708370, 67 ZS555-F40 | US9708370, ZS555-F40) | PDB Reactome pathway UniProtKB/SwissProt GoogleScholar AffyNet | KEGG PC cid PC sid UniChem | US Patent | n/a | n/a | 2.95E+3 | n/a | n/a | n/a | n/a | 7.3 | n/a |
VALORISATION-RECHERCHE, LIMITED PARTNERSHIP; VALORISATION HSJ, LIMITED PARTNERSHIP US Patent | Assay Description Competition experiments were performed by incubating 50 μg of LLC-PK1 membranes expressing human GHS-R1a with 15 fmol of 125I-Ghrelin and increa... | US Patent US9708370 (2017) BindingDB Entry DOI: 10.7270/Q2XP76ZK | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Platelet glycoprotein 4 (Rattus norvegicus) | BDBM263256 (US9708370, 67 ZS555-F40 | US9708370, ZS555-F40) | PDB Reactome pathway UniProtKB/SwissProt GoogleScholar AffyNet | KEGG PC cid PC sid UniChem | Article PubMed | n/a | n/a | 9.19E+3 | n/a | n/a | n/a | n/a | n/a | n/a |
Universit£ de Montr£al Curated by ChEMBL | Assay Description Inhibition of photoactivatable [125I]-Tyr-Bpa-Ala-hexarelin binding to CD36 in Sprague-Dawley rat heart membranes after 60 mins by SDS-PAGE analysis | J Med Chem 60: 9263-9274 (2017) Article DOI: 10.1021/acs.jmedchem.7b01209 BindingDB Entry DOI: 10.7270/Q2GF0WWV | |||||||||||
More data for this Ligand-Target Pair |