Target/Host (Institution) | Ligand | Target/Host Links | Ligand Links | Trg + Lig Links | Ki nM | ΔG° kJ/mole | IC50 nM | Kd nM | EC50/IC50 nM | koff s-1 | kon M-1s-1 | pH | Temp °C |
---|---|---|---|---|---|---|---|---|---|---|---|---|---|
Platelet-derived growth factor receptor beta (Mus musculus (mouse)) | BDBM16590 (2-(1H-indazol-3-yl)-1H-1,3-benzodiazole | 3-(1H-be...) | KEGG UniProtKB/SwissProt GoogleScholar AffyNet | Purchase CHEMBL DrugBank MMDB PC cid PC sid PDB UniChem Patents Similars | Article PubMed | n/a | n/a | 3.40E+3 | n/a | n/a | n/a | n/a | n/a | n/a |
Chiron Corporation Curated by ChEMBL | Assay Description Inhibition of PDGFRbeta | Bioorg Med Chem Lett 16: 3595-9 (2006) Article DOI: 10.1016/j.bmcl.2006.03.069 BindingDB Entry DOI: 10.7270/Q2BZ65N7 | |||||||||||
More data for this Ligand-Target Pair |