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Found 1 hit Enz. Inhib. hit(s) with Target = 'Platelet-derived growth factor receptor beta' and Ligand = 'BDBM3949'   
Target/Host
(Institution)
LigandTarget/Host
Links
Ligand
Links
Trg + Lig
Links
Ki
nM
ΔG°
kJ/mole
IC50
nM
Kd
nM
EC50/IC50
nM
koff
s-1
kon
M-1s-1
pHTemp
°C
Platelet-derived growth factor receptor beta


(Homo sapiens (Human))
BDBM3949
PNG
(5-Methoxy-6-methyl-1-phenylbenzimidazole Hydrochlo...)
Show SMILES COc1cc2ncn(-c3ccccc3)c2cc1C
Show InChI InChI=1S/C15H14N2O/c1-11-8-14-13(9-15(11)18-2)16-10-17(14)12-6-4-3-5-7-12/h3-10H,1-2H3
PDB
MMDB

NCI pathway
Reactome pathway
KEGG

UniProtKB/SwissProt

B.MOAD
DrugBank
antibodypedia
GoogleScholar
AffyNet 
PC cid
PC sid
UniChem

Patents


Similars

Article
PubMed
n/an/a 1.00E+3n/an/an/an/an/an/a



University of Auckland



Assay Description
IC50 is the inhibitor concentration which inhibits 50% of kinase activity that catalyzes the transfer of the terminal phosphate from [gamma-32P] labe...


J Med Chem 42: 2373-82 (1999)


Article DOI: 10.1021/jm980658b
BindingDB Entry DOI: 10.7270/Q2W957B2
More data for this
Ligand-Target Pair