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Compile Data Set for Download or QSAR

Found 1 hit Enz. Inhib. hit(s) with Target = 'Platelet-derived growth factor receptor beta' and Ligand = 'BDBM50132229'   
Target/Host
(Institution)		LigandTarget/Host
Links		Ligand
Links		Trg + Lig
Links		Ki
nM		ΔG°
kJ/mole		IC50
nM		Kd
nM		EC50/IC50
nM		koff
s-1		kon
M-1s-1		pHTemp
°C
Platelet-derived growth factor receptor beta


(Homo sapiens (Human))		BDBM50132229
PNG
(4-(7-Methyl-quinazolin-4-yl)-piperazine-1-carboxyl...)
Show SMILES Cc1ccc2c(ncnc2c1)N1CCN(CC1)C(=O)Nc1ccc(Oc2ccccc2)cc1
Show InChI InChI=1S/C26H25N5O2/c1-19-7-12-23-24(17-19)27-18-28-25(23)30-13-15-31(16-14-30)26(32)29-20-8-10-22(11-9-20)33-21-5-3-2-4-6-21/h2-12,17-18H,13-16H2,1H3,(H,29,32)
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n/an/a>100n/an/an/an/an/an/a



Kyowa Hakko Kogyo Co., Ltd.

Curated by ChEMBL


Assay Description
Inhibitory concentration against platelet-derived growth factor receptor beta phosphorylation in CHO cells

Bioorg Med Chem Lett 13: 3001-4 (2003)


BindingDB Entry DOI: 10.7270/Q2668CKR
More data for this
Ligand-Target Pair