Target/Host (Institution) | Ligand | Target/Host Links | Ligand Links | Trg + Lig Links | Ki nM | ΔG° kJ/mole | IC50 nM | Kd nM | EC50/IC50 nM | koff s-1 | kon M-1s-1 | pH | Temp °C |
---|---|---|---|---|---|---|---|---|---|---|---|---|---|
Potassium voltage-gated channel subfamily B member 1 (Rattus norvegicus) | BDBM50213092 ((1R,2R)-1-(1-naphthalenethoxy)-2-(4-morpholinyl)cy...) | PDB Reactome pathway KEGG UniProtKB/SwissProt GoogleScholar AffyNet | CHEMBL PC cid PC sid UniChem | Article PubMed | n/a | n/a | 3.20E+3 | n/a | n/a | n/a | n/a | n/a | n/a |
Cardiome Pharma Corporation Curated by ChEMBL | Assay Description Inhibition of rat potassium channel Kv2.1 by patch-clamp method | J Med Chem 50: 2818-41 (2007) Article DOI: 10.1021/jm0604528 BindingDB Entry DOI: 10.7270/Q29Z95QZ | |||||||||||
More data for this Ligand-Target Pair |