Target/Host (Institution) | Ligand | Target/Host Links | Ligand Links | Trg + Lig Links | Ki nM | ΔG° kJ/mole | IC50 nM | Kd nM | EC50/IC50 nM | koff s-1 | kon M-1s-1 | pH | Temp °C |
---|---|---|---|---|---|---|---|---|---|---|---|---|---|
Potassium voltage-gated channel subfamily H member 2 (Homo sapiens (Human)) | BDBM50275432 (CHEMBL487965 | S-2-(6-(1,4-dihydrobenzo[d][1,2]dio...) | PDB MMDB Reactome pathway KEGG UniProtKB/SwissProt UniProtKB/TrEMBL B.MOAD DrugBank antibodypedia GoogleScholar AffyNet | CHEMBL KEGG PC cid PC sid UniChem | Article PubMed | n/a | n/a | n/a | n/a | >3.00E+4 | n/a | n/a | n/a | n/a |
Kalypsys, Inc. Curated by ChEMBL | Assay Description Inhibition of human ERG by patch-clamp assay | Bioorg Med Chem Lett 18: 6093-6 (2008) Article DOI: 10.1016/j.bmcl.2008.10.029 BindingDB Entry DOI: 10.7270/Q2F18ZJS | |||||||||||
More data for this Ligand-Target Pair |