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Compile Data Set for Download or QSAR

Found 1 hit Enz. Inhib. hit(s) with Target = 'Progesterone receptor' and Ligand = 'BDBM50290375'   
Target/Host
(Institution)
LigandTarget/Host
Links
Ligand
Links
Trg + Lig
Links
Ki
nM
ΔG°
kJ/mole
IC50
nM
Kd
nM
EC50/IC50
nM
koff
s-1
kon
M-1s-1
pHTemp
°C
Progesterone receptor


(Oryctolagus cuniculus)
BDBM50290375
PNG
(CHEMBL314154 | N-[1-[1-(4-Fluoro-phenyl)-7-naphtha...)
Show SMILES CN=NCc1nn(c2C(Cc3cccc4ccccc34)CCCc12)-c1ccc(F)cc1 |w:1.0|
Show InChI InChI=1S/C26H25FN4/c1-28-29-17-25-24-11-5-9-20(16-19-8-4-7-18-6-2-3-10-23(18)19)26(24)31(30-25)22-14-12-21(27)13-15-22/h2-4,6-8,10,12-15,20H,5,9,11,16-17H2,1H3
PDB
MMDB

KEGG

UniProtKB/SwissProt

B.MOAD
GoogleScholar
AffyNet 
CHEMBL
PC cid
PC sid
UniChem
Article
n/an/a 49n/an/an/an/an/an/a



TBA

Curated by ChEMBL


Assay Description
Binding affinity determined by ability to displace [3H]-R5020 radioligand using uterine progesterone receptor obtained from estrogen-primed rabbit


Bioorg Med Chem Lett 7: 2551-2556 (1997)


Article DOI: 10.1016/S0960-894X(97)10016-6
BindingDB Entry DOI: 10.7270/Q2MW2H5C
More data for this
Ligand-Target Pair