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Found 1 hit Enz. Inhib. hit(s) with Target = 'Protein arginine N-methyltransferase 3' and Ligand = 'BDBM50247353'   
Target/Host
(Institution)		LigandTarget/Host
Links		Ligand
Links		Trg + Lig
Links		Ki
nM		ΔG°
kJ/mole		IC50
nM		Kd
nM		EC50/IC50
nM		koff
s-1		kon
M-1s-1		pHTemp
°C
Protein arginine N-methyltransferase 3


(Homo sapiens)		BDBM50247353
PNG
(CHEMBL4081032)
Show SMILES O=C(NCCC1CCCC1)Nc1ccc2cnccc2c1
Show InChI InChI=1S/C17H21N3O/c21-17(19-10-7-13-3-1-2-4-13)20-16-6-5-15-12-18-9-8-14(15)11-16/h5-6,8-9,11-13H,1-4,7,10H2,(H2,19,20,21)
PDB

UniProtKB/SwissProt

antibodypedia
GoogleScholar
AffyNet 
PC cid
PC sid
UniChem

Similars
Article
PubMed
n/an/a 295n/an/an/an/an/an/a



Icahn School of Medicine at Mount Sinai

Curated by ChEMBL


Assay Description
Inhibition of PRMT3 (unknown origin) using C-terminally biotinylated histone H4 as substrate in presence of [3H]S-adenosylmethionine by scintillation...

J Med Chem 61: 1204-1217 (2018)


Article DOI: 10.1021/acs.jmedchem.7b01674
BindingDB Entry DOI: 10.7270/Q24J0HK6
More data for this
Ligand-Target Pair