BindingDB PrimarySearch

Found 2 hits Enz. Inhib. hit(s) with Target = 'Protein kinase C alpha type' and Ligand = 'BDBM50087240'
Target/Host (Institution)	Ligand	Target/Host Links	Ligand Links	Trg + Lig Links	Ki nM	ΔG° kJ/mole	IC50 nM	Kd nM	EC50/IC50 nM	k_off s^-1	k_on M^-1s^-1	pH	Temp °C
Protein kinase C alpha type (Homo sapiens (Human))	BDBM50087240 ((E)-Octadec-9-enoic acid (S)-1-hydroxymethyl-2-((E...) Show SMILES Show InChI	PDB MMDB NCI pathway Reactome pathway KEGG UniProtKB/SwissProt B.MOAD DrugBank antibodypedia GoogleScholar AffyNet	Purchase CHEMBL KEGG PC cid PC sid UniChem Similars	PubMed	87	n/a	n/a	n/a	n/a	n/a	n/a	n/a	n/a
National Cancer Institute Curated by ChEMBL					Assay Description Displacement of [20-3H] phorbol 12,13-dibutyrate from protein kinase C alpha				Bioorg Med Chem Lett 10: 653-5 (2000) BindingDB Entry DOI: 10.7270/Q2G16011
National Cancer Institute Curated by ChEMBL					More data for this Ligand-Target Pair
Protein kinase C alpha type (Bos taurus (bovine))	BDBM50087240 ((E)-Octadec-9-enoic acid (S)-1-hydroxymethyl-2-((E...) Show SMILES Show InChI	PDB MMDB Reactome pathway KEGG UniProtKB/SwissProt B.MOAD GoogleScholar AffyNet	Purchase CHEMBL KEGG PC cid PC sid UniChem Similars	PubMed	87.2	n/a	n/a	n/a	n/a	n/a	n/a	n/a	n/a
National Cancer Institute at Frederick Curated by ChEMBL					Assay Description Ability to displace bound [20-3H]-PDBU from a recombinant single isozyme (PKCalpha) in the presence of phosphatidylserine				J Med Chem 44: 1892-904 (2001) BindingDB Entry DOI: 10.7270/Q2H995WH
National Cancer Institute at Frederick Curated by ChEMBL					More data for this Ligand-Target Pair