BindingDB PrimarySearch

Found 7 hits Enz. Inhib. hit(s) with Target = 'Protein kinase C delta type' and Ligand = 'BDBM50057509'
Target/Host (Institution)	Ligand	Target/Host Links	Ligand Links	Trg + Lig Links	Ki nM	ΔG° kJ/mole	IC50 nM	Kd nM	EC50/IC50 nM	k_off s^-1	k_on M^-1s^-1	pH	Temp °C
Protein kinase C delta type (Mus musculus)	BDBM50057509 ((2S,5S)-8-Dec-1-ynyl-5-hydroxymethyl-2-isopropyl-1...) Show SMILES Show InChI	PDB MMDB Reactome pathway KEGG UniProtKB/SwissProt B.MOAD DrugBank GoogleScholar AffyNet	CHEMBL PC cid PC sid UniChem Patents Similars	PubMed	10.7	n/a	n/a	n/a	n/a	n/a	n/a	n/a	n/a
Georgetown University Medical Center Curated by ChEMBL					Assay Description Displacement of [3H]- PDBu from Protein kinase C delta C1b domain				J Med Chem 45: 853-60 (2002) BindingDB Entry DOI: 10.7270/Q20C4V25
Georgetown University Medical Center Curated by ChEMBL					More data for this Ligand-Target Pair
Protein kinase C delta type (Homo sapiens (Human))	BDBM50057509 ((2S,5S)-8-Dec-1-ynyl-5-hydroxymethyl-2-isopropyl-1...) Show SMILES Show InChI	PDB MMDB NCI pathway Reactome pathway KEGG UniProtKB/SwissProt B.MOAD DrugBank antibodypedia GoogleScholar AffyNet	CHEMBL PC cid PC sid UniChem Patents Similars	Article PubMed	11	n/a	n/a	n/a	n/a	n/a	n/a	n/a	n/a
Georgetown University Medical Center Curated by ChEMBL					Assay Description Inhibition of [3H]-PDBu binding to PKC delta wild type				J Med Chem 40: 1316-26 (1997) Article DOI: 10.1021/jm960875h BindingDB Entry DOI: 10.7270/Q2319TZS
Georgetown University Medical Center Curated by ChEMBL					More data for this Ligand-Target Pair
Protein kinase C delta type (Homo sapiens (Human))	BDBM50057509 ((2S,5S)-8-Dec-1-ynyl-5-hydroxymethyl-2-isopropyl-1...) Show SMILES Show InChI	PDB MMDB NCI pathway Reactome pathway KEGG UniProtKB/SwissProt B.MOAD DrugBank antibodypedia GoogleScholar AffyNet	CHEMBL PC cid PC sid UniChem Patents Similars	PubMed	114	n/a	n/a	n/a	n/a	n/a	n/a	n/a	n/a
Georgetotwn University Curated by ChEMBL					Assay Description Inhibition of [3H]-phorbol 12,13-dibutyrate (PDBu) binding to human recombinant protein kinase C delta				Bioorg Med Chem Lett 11: 955-9 (2001) BindingDB Entry DOI: 10.7270/Q2D799PV
Georgetotwn University Curated by ChEMBL					More data for this Ligand-Target Pair
Protein kinase C delta type (Homo sapiens (Human))	BDBM50057509 ((2S,5S)-8-Dec-1-ynyl-5-hydroxymethyl-2-isopropyl-1...) Show SMILES Show InChI	PDB MMDB NCI pathway Reactome pathway KEGG UniProtKB/SwissProt B.MOAD DrugBank antibodypedia GoogleScholar AffyNet	CHEMBL PC cid PC sid UniChem Patents Similars	Article PubMed	122	n/a	n/a	n/a	n/a	n/a	n/a	n/a	n/a
Georgetown University Medical Center Curated by ChEMBL					Assay Description Displacement of [3H]- PDBu from recombinant PKC delta expressed in baculovirus				J Med Chem 40: 1316-26 (1997) Article DOI: 10.1021/jm960875h BindingDB Entry DOI: 10.7270/Q2319TZS
Georgetown University Medical Center Curated by ChEMBL					More data for this Ligand-Target Pair
Protein kinase C delta type (Homo sapiens (Human))	BDBM50057509 ((2S,5S)-8-Dec-1-ynyl-5-hydroxymethyl-2-isopropyl-1...) Show SMILES Show InChI	PDB MMDB NCI pathway Reactome pathway KEGG UniProtKB/SwissProt B.MOAD DrugBank antibodypedia GoogleScholar AffyNet	CHEMBL PC cid PC sid UniChem Patents Similars	Article PubMed	134	n/a	n/a	n/a	n/a	n/a	n/a	n/a	n/a
Georgetown University Medical Center Curated by ChEMBL					Assay Description Inhibition of [3H]-PDBu binding to PKC delta mutant Leu 20-Gly				J Med Chem 40: 1316-26 (1997) Article DOI: 10.1021/jm960875h BindingDB Entry DOI: 10.7270/Q2319TZS
Georgetown University Medical Center Curated by ChEMBL					More data for this Ligand-Target Pair
Protein kinase C delta type (Homo sapiens (Human))	BDBM50057509 ((2S,5S)-8-Dec-1-ynyl-5-hydroxymethyl-2-isopropyl-1...) Show SMILES Show InChI	PDB MMDB NCI pathway Reactome pathway KEGG UniProtKB/SwissProt B.MOAD DrugBank antibodypedia GoogleScholar AffyNet	CHEMBL PC cid PC sid UniChem Patents Similars	Article PubMed	730	n/a	n/a	n/a	n/a	n/a	n/a	n/a	n/a
Georgetown University Medical Center Curated by ChEMBL					Assay Description Inhibition of [3H]-PDBu binding to PKC delta mutant Pro 11-Gly				J Med Chem 40: 1316-26 (1997) Article DOI: 10.1021/jm960875h BindingDB Entry DOI: 10.7270/Q2319TZS
Georgetown University Medical Center Curated by ChEMBL					More data for this Ligand-Target Pair
Protein kinase C delta type (Homo sapiens (Human))	BDBM50057509 ((2S,5S)-8-Dec-1-ynyl-5-hydroxymethyl-2-isopropyl-1...) Show SMILES Show InChI	PDB MMDB NCI pathway Reactome pathway KEGG UniProtKB/SwissProt B.MOAD DrugBank antibodypedia GoogleScholar AffyNet	CHEMBL PC cid PC sid UniChem Patents Similars	Article PubMed	933	n/a	n/a	n/a	n/a	n/a	n/a	n/a	n/a
Georgetown University Medical Center Curated by ChEMBL					Assay Description Inhibition of [3H]-PDBu binding to PKC delta mutant Gln 27-Val				J Med Chem 40: 1316-26 (1997) Article DOI: 10.1021/jm960875h BindingDB Entry DOI: 10.7270/Q2319TZS
Georgetown University Medical Center Curated by ChEMBL					More data for this Ligand-Target Pair