Target/Host (Institution) | Ligand | Target/Host Links | Ligand Links | Trg + Lig Links | Ki nM | ΔG° kJ/mole | IC50 nM | Kd nM | EC50/IC50 nM | koff s-1 | kon M-1s-1 | pH | Temp °C |
---|---|---|---|---|---|---|---|---|---|---|---|---|---|
Protein-glutamine gamma-glutamyltransferase 2 (Mus musculus) | BDBM50392906 (CHEMBL2152204) | KEGG UniProtKB/SwissProt GoogleScholar AffyNet | CHEMBL PC cid PC sid UniChem Similars | Article PubMed | n/a | n/a | 55 | n/a | n/a | n/a | n/a | n/a | n/a |
TBA Curated by ChEMBL | Assay Description Inhibition of mouse TGM2 | ACS Med Chem Lett 3: 731-735 (2012) Article DOI: 10.1021/ml3001352 BindingDB Entry DOI: 10.7270/Q2Q241B7 | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Protein-glutamine gamma-glutamyltransferase 2 (Homo sapiens (Human)) | BDBM50392906 (CHEMBL2152204) | PDB MMDB KEGG UniProtKB/SwissProt B.MOAD DrugBank antibodypedia GoogleScholar AffyNet | CHEMBL PC cid PC sid UniChem Similars | Article PubMed | n/a | n/a | 110 | n/a | n/a | n/a | n/a | n/a | n/a |
TBA Curated by ChEMBL | Assay Description Inhibition of human TGM2 | ACS Med Chem Lett 3: 731-735 (2012) Article DOI: 10.1021/ml3001352 BindingDB Entry DOI: 10.7270/Q2Q241B7 | |||||||||||
More data for this Ligand-Target Pair |