Target/Host (Institution) | Ligand | Target/Host Links | Ligand Links | Trg + Lig Links | Ki nM | ΔG° kJ/mole | IC50 nM | Kd nM | EC50/IC50 nM | koff s-1 | kon M-1s-1 | pH | Temp °C |
---|---|---|---|---|---|---|---|---|---|---|---|---|---|
Receptor tyrosine-protein kinase erbB-2 (Homo sapiens (Human)) | BDBM50210879 (CHEMBL3218531) | PDB MMDB UniProtKB/SwissProt B.MOAD DrugBank antibodypedia GoogleScholar AffyNet | CHEMBL PC cid PC sid UniChem Similars | Article PubMed | n/a | n/a | n/a | 1.00E+3 | n/a | n/a | n/a | n/a | n/a |
University of Louisiana at Monroe Curated by ChEMBL | Assay Description Binding affinity to HER2 extracellular domain (unknown origin) by SPR assay | Eur J Med Chem 125: 914-924 (2017) Article DOI: 10.1016/j.ejmech.2016.10.015 BindingDB Entry DOI: 10.7270/Q2PR7Z4F | |||||||||||
More data for this Ligand-Target Pair |