Target/Host (Institution) | Ligand | Target/Host Links | Ligand Links | Trg + Lig Links | Ki nM | ΔG° kJ/mole | IC50 nM | Kd nM | EC50/IC50 nM | koff s-1 | kon M-1s-1 | pH | Temp °C |
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Ribosomal protein S6 kinase alpha-3 (Homo sapiens (Human)) | BDBM50381082 (CHEMBL2017521) | PDB MMDB Reactome pathway KEGG UniProtKB/SwissProt B.MOAD DrugBank antibodypedia GoogleScholar AffyNet | CHEMBL PC cid PC sid UniChem Similars | Article PubMed | n/a | n/a | 493 | n/a | n/a | n/a | n/a | n/a | n/a |
University of Virginia Curated by ChEMBL | Assay Description Inhibition of His-tagged RSK2 expressed in Sf9 cells using ERalpha-Ser167 RLASTND as substrate after 120 mins by chemiluminescence assay | Bioorg Med Chem Lett 22: 3244-7 (2012) Article DOI: 10.1016/j.bmcl.2012.03.033 BindingDB Entry DOI: 10.7270/Q2QN67S5 | |||||||||||
More data for this Ligand-Target Pair | 3D Structure (docked) |