Target/Host (Institution) | Ligand | Target/Host Links | Ligand Links | Trg + Lig Links | Ki nM | ΔG° kJ/mole | IC50 nM | Kd nM | EC50/IC50 nM | koff s-1 | kon M-1s-1 | pH | Temp °C |
---|---|---|---|---|---|---|---|---|---|---|---|---|---|
Serine/threonine-protein kinase B-raf (Homo sapiens (Human)) | BDBM50121690 (CHEMBL3616960) | PDB MMDB NCI pathway Reactome pathway KEGG UniProtKB/SwissProt B.MOAD DrugBank antibodypedia GoogleScholar AffyNet | CHEMBL PC cid PC sid UniChem | Article PubMed | n/a | n/a | 668 | n/a | n/a | n/a | n/a | n/a | n/a |
Hanyang University Curated by ChEMBL | Assay Description Inhibition of BRAF V599E mutant (unknown origin) after 40 mins by scintillation counting analysis | Eur J Med Chem 102: 600-10 (2015) Article DOI: 10.1016/j.ejmech.2015.08.031 BindingDB Entry DOI: 10.7270/Q2XG9SXV | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Serine/threonine-protein kinase B-raf (Homo sapiens (Human)) | BDBM50121690 (CHEMBL3616960) | PDB MMDB NCI pathway Reactome pathway KEGG UniProtKB/SwissProt B.MOAD DrugBank antibodypedia GoogleScholar AffyNet | CHEMBL PC cid PC sid UniChem | Article PubMed | n/a | n/a | 5.96E+3 | n/a | n/a | n/a | n/a | n/a | n/a |
Hanyang University Curated by ChEMBL | Assay Description Inhibition of BRAF (unknown origin) after 40 mins by scintillation counting analysis | Eur J Med Chem 102: 600-10 (2015) Article DOI: 10.1016/j.ejmech.2015.08.031 BindingDB Entry DOI: 10.7270/Q2XG9SXV | |||||||||||
More data for this Ligand-Target Pair |