Target/Host (Institution) | Ligand | Target/Host Links | Ligand Links | Trg + Lig Links | Ki nM | ΔG° kJ/mole | IC50 nM | Kd nM | EC50/IC50 nM | koff s-1 | kon M-1s-1 | pH | Temp °C |
---|---|---|---|---|---|---|---|---|---|---|---|---|---|
Serine/threonine-protein kinase Nek2 (Homo sapiens (Human)) | BDBM50441090 (CHEMBL2430323 | US9669028, 114 N-(3-(3-methyl-1H-p...) | PDB UniProtKB/SwissProt antibodypedia GoogleScholar AffyNet | Purchase CHEMBL MCE PC cid PC sid UniChem | Article PubMed | n/a | n/a | 2.00E+3 | n/a | n/a | n/a | n/a | n/a | n/a |
University of Edinburgh Cancer Research Centre in the Institute of Genetics and Molecular Medicine Curated by ChEMBL | Assay Description Inhibition of human NEK2alpha in presence of 50 uM ATP | Bioorg Med Chem Lett 23: 5578-85 (2013) Article DOI: 10.1016/j.bmcl.2013.08.046 BindingDB Entry DOI: 10.7270/Q2Q52R2M | |||||||||||
More data for this Ligand-Target Pair |