Target/Host (Institution) | Ligand | Target/Host Links | Ligand Links | Trg + Lig Links | Ki nM | ΔG° kJ/mole | IC50 nM | Kd nM | EC50/IC50 nM | koff s-1 | kon M-1s-1 | pH | Temp °C |
---|---|---|---|---|---|---|---|---|---|---|---|---|---|
Serine/threonine-protein kinase PLK1 (Homo sapiens (Human)) | BDBM47167 (CHEMBL201511 | US8957103, Z1 | US9364459, A) | PDB MMDB NCI pathway Reactome pathway KEGG UniProtKB/SwissProt B.MOAD DrugBank antibodypedia GoogleScholar AffyNet | CHEMBL PC cid PC sid UniChem Similars | Article PubMed | n/a | n/a | >1.00E+5 | n/a | n/a | n/a | n/a | n/a | n/a |
Eberhard Karls University Curated by ChEMBL | Assay Description Inhibition of human PLK1 | J Med Chem 49: 7549-53 (2006) Article DOI: 10.1021/jm0609871 BindingDB Entry DOI: 10.7270/Q2NZ8794 | |||||||||||
More data for this Ligand-Target Pair |