Target/Host (Institution) | Ligand | Target/Host Links | Ligand Links | Trg + Lig Links | Ki nM | ΔG° kJ/mole | IC50 nM | Kd nM | EC50/IC50 nM | koff s-1 | kon M-1s-1 | pH | Temp °C |
---|---|---|---|---|---|---|---|---|---|---|---|---|---|
Serine/threonine-protein kinase pim-1 (Homo sapiens (Human)) | BDBM110767 (US8614206, 316 | US8614206, 317 | US8614206, 320 |...) | PDB MMDB KEGG UniProtKB/SwissProt B.MOAD DrugBank antibodypedia GoogleScholar AffyNet | PC cid PC sid UniChem Similars | US Patent | 0.00700 | n/a | n/a | n/a | n/a | n/a | n/a | 7.2 | n/a |
F. Hoffmann-La Roche AG US Patent | Assay Description PIM-1, -2, and -3 enzymes were generated as fusion proteins expressed in bacteria and purified by IMAC column chromatography (Sun, X., Chiu, J. F., a... | US Patent US8614206 (2013) BindingDB Entry DOI: 10.7270/Q2W66JFG | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Serine/threonine-protein kinase pim-1 (Homo sapiens (Human)) | BDBM110767 (US8614206, 316 | US8614206, 317 | US8614206, 320 |...) | PDB MMDB KEGG UniProtKB/SwissProt B.MOAD DrugBank antibodypedia GoogleScholar AffyNet | PC cid PC sid UniChem Similars | US Patent | 0.0180 | n/a | n/a | n/a | n/a | n/a | n/a | 7.2 | n/a |
F. Hoffmann-La Roche AG US Patent | Assay Description PIM-1, -2, and -3 enzymes were generated as fusion proteins expressed in bacteria and purified by IMAC column chromatography (Sun, X., Chiu, J. F., a... | US Patent US8614206 (2013) BindingDB Entry DOI: 10.7270/Q2W66JFG | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Serine/threonine-protein kinase pim-1 (Homo sapiens (Human)) | BDBM110767 (US8614206, 316 | US8614206, 317 | US8614206, 320 |...) | PDB MMDB KEGG UniProtKB/SwissProt B.MOAD DrugBank antibodypedia GoogleScholar AffyNet | PC cid PC sid UniChem Similars | US Patent | 0.0500 | n/a | n/a | n/a | n/a | n/a | n/a | 7.2 | n/a |
F. Hoffmann-La Roche AG US Patent | Assay Description PIM-1, -2, and -3 enzymes were generated as fusion proteins expressed in bacteria and purified by IMAC column chromatography (Sun, X., Chiu, J. F., a... | US Patent US8614206 (2013) BindingDB Entry DOI: 10.7270/Q2W66JFG | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Serine/threonine-protein kinase pim-1 (Homo sapiens (Human)) | BDBM110767 (US8614206, 316 | US8614206, 317 | US8614206, 320 |...) | PDB MMDB KEGG UniProtKB/SwissProt B.MOAD DrugBank antibodypedia GoogleScholar AffyNet | PC cid PC sid UniChem Similars | US Patent | 0.0970 | n/a | n/a | n/a | n/a | n/a | n/a | 7.2 | n/a |
F. Hoffmann-La Roche AG US Patent | Assay Description PIM-1, -2, and -3 enzymes were generated as fusion proteins expressed in bacteria and purified by IMAC column chromatography (Sun, X., Chiu, J. F., a... | US Patent US8614206 (2013) BindingDB Entry DOI: 10.7270/Q2W66JFG | |||||||||||
More data for this Ligand-Target Pair |