Compile Data Set for Download or QSAR

Found 1 hit Enz. Inhib. hit(s) with Target = 'Serine/threonine-protein kinase pim-1' and Ligand = 'BDBM50021654'   

Target/Host (Institution)	Ligand	Target/Host Links	Ligand Links	Trg + Lig Links	Ki nM	ΔG° kJ/mole	IC50 nM	Kd nM	EC50/IC50 nM	koff s-1	kon M-1s-1	pH	Temp °C
Serine/threonine-protein kinase pim-1 (Homo sapiens (Human))	BDBM50021654 (CHEMBL3297760) Show SMILES CN1CCN([C@H](C1)c1ccccc1)C(=O)C[C@H]1CNC(=O)c2cc(cn12)-c1cccc(F)c1 |r| Show InChI InChI=1S/C26H27FN4O2/c1-29-10-11-30(24(17-29)18-6-3-2-4-7-18)25(32)14-22-15-28-26(33)23-13-20(16-31(22)23)19-8-5-9-21(27)12-19/h2-9,12-13,16,22,24H,10-11,14-15,17H2,1H3,(H,28,33)/t22-,24+/m0/s1	PDB MMDB KEGG UniProtKB/SwissProt B.MOAD DrugBank antibodypedia GoogleScholar AffyNet	CHEMBL PC cid PC sid UniChem Patents Similars	Article PubMed	n/a	n/a	233	n/a	n/a	n/a	n/a	n/a	n/a
Nerviano Medical Sciences Curated by ChEMBL					Assay Description Inhibition of human PIM1 using ARK-RERTYSFGHHA as substrate incubated for 60 mins prior to substrate addition by topcount scintillation counting anal...				Bioorg Med Chem 21: 7364-80 (2013) Article DOI: 10.1016/j.bmc.2013.09.054 BindingDB Entry DOI: 10.7270/Q23F4R7S
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