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Found 1 hit Enz. Inhib. hit(s) with Target = 'Serine/threonine-protein kinase pim-3' and Ligand = 'BDBM50326438'   
Target/Host
(Institution)
LigandTarget/Host
Links
Ligand
Links
Trg + Lig
Links
Ki
nM
ΔG°
kJ/mole
IC50
nM
Kd
nM
EC50/IC50
nM
koff
s-1
kon
M-1s-1
pHTemp
°C
Serine/threonine-protein kinase pim-3


(Homo sapiens (Human))
BDBM50326438
PNG
(9-trifluoromethyl-1,10-dihydropyrrolo[2,3-a]carbaz...)
Show SMILES FC(F)(F)c1cccc2c1[nH]c1c2ccc2c(C=O)c[nH]c12
Show InChI InChI=1S/C16H9F3N2O/c17-16(18,19)12-3-1-2-10-11-5-4-9-8(7-22)6-20-14(9)15(11)21-13(10)12/h1-7,20-21H
KEGG

UniProtKB/SwissProt

antibodypedia
GoogleScholar
AffyNet 
CHEMBL
PC cid
PC sid
UniChem
Article
PubMed
n/an/a 6n/an/an/an/an/an/a



Clermont Université

Curated by ChEMBL


Assay Description
Inhibition of human GST fused Pim3 expressed in Escherichia coli after 30 mins


Bioorg Med Chem 18: 6865-73 (2010)


Article DOI: 10.1016/j.bmc.2010.07.036
BindingDB Entry DOI: 10.7270/Q2PK0GBZ
More data for this
Ligand-Target Pair