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Found 1 hit Enz. Inhib. hit(s) with Target = 'Serine/threonine-protein kinase pim-3' and Ligand = 'BDBM50432942'   
Target/Host
(Institution)
LigandTarget/Host
Links
Ligand
Links
Trg + Lig
Links
Ki
nM
ΔG°
kJ/mole
IC50
nM
Kd
nM
EC50/IC50
nM
koff
s-1
kon
M-1s-1
pHTemp
°C
Serine/threonine-protein kinase pim-3


(Homo sapiens (Human))
BDBM50432942
PNG
(CHEMBL2377721)
Show SMILES Nc1cc2cn[nH]c2c2cc[nH]c12
Show InChI InChI=1S/C9H8N4/c10-7-3-5-4-12-13-8(5)6-1-2-11-9(6)7/h1-4,11H,10H2,(H,12,13)
KEGG

UniProtKB/SwissProt

antibodypedia
GoogleScholar
AffyNet 
CHEMBL
PC cid
PC sid
UniChem
Article
PubMed
n/an/a 33n/an/an/an/an/an/a



Clermont Universit£

Curated by ChEMBL


Assay Description
Inhibition of human full length Pim-3 using RSRHSSYPAGT as substrate assessed as residual activity after 30 mins in presence of [gamma-33P]ATP


Bioorg Med Chem Lett 23: 2298-301 (2013)


Article DOI: 10.1016/j.bmcl.2013.02.074
BindingDB Entry DOI: 10.7270/Q26111PK
More data for this
Ligand-Target Pair