Target/Host (Institution) | Ligand | Target/Host Links | Ligand Links | Trg + Lig Links | Ki nM | ΔG° kJ/mole | IC50 nM | Kd nM | EC50/IC50 nM | koff s-1 | kon M-1s-1 | pH | Temp °C |
---|---|---|---|---|---|---|---|---|---|---|---|---|---|
Sigma non-opioid intracellular receptor 1 (Homo sapiens (Human)) | BDBM50061754 (CHEMBL542487 | N-(2-Chloro-3,5-diethyl-phenyl)-N'-...) | PDB UniProtKB/SwissProt antibodypedia GoogleScholar AffyNet | CHEMBL PC cid PC sid UniChem Similars | Article PubMed | n/a | n/a | 4.5 | n/a | n/a | n/a | n/a | n/a | n/a |
Cambridge NeuroScience, Inc. Curated by ChEMBL | Assay Description Binding assay for the sigma receptor sites is performed by utilizing [3H]N,N-di-o-tolylguanidine ([3H]DTG) and guinea pig brain membrane suspensions | J Med Chem 40: 4281-9 (1998) Article DOI: 10.1021/jm970459c BindingDB Entry DOI: 10.7270/Q2G161HQ | |||||||||||
More data for this Ligand-Target Pair |