Target/Host (Institution) | Ligand | Target/Host Links | Ligand Links | Trg + Lig Links | Ki nM | ΔG° kJ/mole | IC50 nM | Kd nM | EC50/IC50 nM | koff s-1 | kon M-1s-1 | pH | Temp °C |
---|---|---|---|---|---|---|---|---|---|---|---|---|---|
Sigma non-opioid intracellular receptor 1 (Homo sapiens (Human)) | BDBM50063805 (6-Benzoyl-3-(2-pyrrolidin-1-yl-ethyl)-3H-benzothia...) | PDB UniProtKB/SwissProt antibodypedia GoogleScholar AffyNet | CHEMBL PC cid PC sid UniChem Similars | Article PubMed | 54 | n/a | n/a | n/a | n/a | n/a | n/a | n/a | n/a |
University of Louvain Curated by ChEMBL | Assay Description The compound was tested for the affinity on sigma 1 receptor using [3H]- pentazocine as radioligand | J Med Chem 41: 1138-45 (1998) Article DOI: 10.1021/jm970682+ BindingDB Entry DOI: 10.7270/Q29S1Q5N | |||||||||||
More data for this Ligand-Target Pair |