Target/Host (Institution) | Ligand | Target/Host Links | Ligand Links | Trg + Lig Links | Ki nM | ΔG° kJ/mole | IC50 nM | Kd nM | EC50/IC50 nM | koff s-1 | kon M-1s-1 | pH | Temp °C |
---|---|---|---|---|---|---|---|---|---|---|---|---|---|
Sigma non-opioid intracellular receptor 1 (Homo sapiens (Human)) | BDBM50065135 (4-Iodo-N-(2-pyrrolidin-1-yl-ethyl)-benzenesulfonam...) | PDB UniProtKB/SwissProt antibodypedia GoogleScholar AffyNet | Purchase CHEMBL PC cid PC sid UniChem Patents Similars | Article PubMed | 1.46 | n/a | n/a | n/a | n/a | n/a | n/a | n/a | n/a |
The George Washington University Medical Center Curated by ChEMBL | Assay Description Inhibition Constant for 4-[125I]-IPBS binding to sigma 1 receptor in guinea pig brain membranes | J Med Chem 41: 2445-50 (1998) Article DOI: 10.1021/jm9800447 BindingDB Entry DOI: 10.7270/Q27P8XHM | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Sigma non-opioid intracellular receptor 1 (Homo sapiens (Human)) | BDBM50065135 (4-Iodo-N-(2-pyrrolidin-1-yl-ethyl)-benzenesulfonam...) | PDB UniProtKB/SwissProt antibodypedia GoogleScholar AffyNet | Purchase CHEMBL PC cid PC sid UniChem Patents Similars | Article PubMed | 4.30 | n/a | n/a | n/a | n/a | n/a | n/a | n/a | n/a |
The George Washington University Medical Center Curated by ChEMBL | Assay Description Inhibition of [3H]-(+)-pentazocine binding to sigma-1 receptor in guinea pig brain membranes | J Med Chem 41: 2445-50 (1998) Article DOI: 10.1021/jm9800447 BindingDB Entry DOI: 10.7270/Q27P8XHM | |||||||||||
More data for this Ligand-Target Pair |