Target/Host (Institution) | Ligand | Target/Host Links | Ligand Links | Trg + Lig Links | Ki nM | ΔG° kJ/mole | IC50 nM | Kd nM | EC50/IC50 nM | koff s-1 | kon M-1s-1 | pH | Temp °C |
---|---|---|---|---|---|---|---|---|---|---|---|---|---|
Sigma non-opioid intracellular receptor 1 (Homo sapiens (Human)) | BDBM50283400 ((1-Benzyl-piperidin-4-yl)-methyl-((E)-3-phenyl-all...) | PDB UniProtKB/SwissProt antibodypedia GoogleScholar AffyNet | CHEMBL PC cid PC sid UniChem Similars | Article | 2.60 | n/a | n/a | n/a | n/a | n/a | n/a | n/a | n/a |
TBA Curated by ChEMBL | Assay Description Inhibiton of [3H]-(+)-SKF-10,047 binding to sigma receptor | Bioorg Med Chem Lett 4: 329-334 (1994) Article DOI: 10.1016/S0960-894X(01)80138-4 BindingDB Entry DOI: 10.7270/Q20R9PBC | |||||||||||
More data for this Ligand-Target Pair |