Target/Host (Institution) | Ligand | Target/Host Links | Ligand Links | Trg + Lig Links | Ki nM | ΔG° kJ/mole | IC50 nM | Kd nM | EC50/IC50 nM | koff s-1 | kon M-1s-1 | pH | Temp °C |
---|---|---|---|---|---|---|---|---|---|---|---|---|---|
Sodium-dependent dopamine transporter (Homo sapiens (Human)) | BDBM50363762 (CHEMBL1947088) | NCI pathway Reactome pathway KEGG UniProtKB/SwissProt DrugBank GoogleScholar AffyNet | CHEMBL PC cid PC sid UniChem Similars | Article PubMed | 0.870 | n/a | n/a | n/a | n/a | n/a | n/a | n/a | n/a |
INSERM Curated by ChEMBL | Assay Description Displacement of [3H]WIN35428 from human cloned DAT receptor expressed in human HEK293 cells | Bioorg Med Chem 20: 1388-95 (2012) Article DOI: 10.1016/j.bmc.2012.01.014 BindingDB Entry DOI: 10.7270/Q26T0N3Z | |||||||||||
More data for this Ligand-Target Pair |