Target/Host (Institution) | Ligand | Target/Host Links | Ligand Links | Trg + Lig Links | Ki nM | ΔG° kJ/mole | IC50 nM | Kd nM | EC50/IC50 nM | koff s-1 | kon M-1s-1 | pH | Temp °C |
---|---|---|---|---|---|---|---|---|---|---|---|---|---|
Somatostatin receptor type 3 (Homo sapiens (Human)) | BDBM50065452 (2-Amino-N-{4-[(2S,5S,8S,14S,17R)-8,14-dibenzyl-5-(...) | Reactome pathway KEGG UniProtKB/SwissProt DrugBank antibodypedia GoogleScholar AffyNet | CHEMBL PC cid PC sid UniChem Similars | Article PubMed | 797 | n/a | n/a | n/a | n/a | n/a | n/a | n/a | n/a |
University of California at San Diego Curated by ChEMBL | Assay Description In vitro inhibition of radioligand binding to human somatostatin receptor (hsst3) expressed in CHO-K1 cells. | J Med Chem 41: 2679-85 (1998) Article DOI: 10.1021/jm970393l BindingDB Entry DOI: 10.7270/Q2Z60N6X | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Somatostatin receptor type 3 (Homo sapiens (Human)) | BDBM50065452 (2-Amino-N-{4-[(2S,5S,8S,14S,17R)-8,14-dibenzyl-5-(...) | Reactome pathway KEGG UniProtKB/SwissProt DrugBank antibodypedia GoogleScholar AffyNet | CHEMBL PC cid PC sid UniChem Similars | Article PubMed | n/a | n/a | n/a | 339 | n/a | n/a | n/a | n/a | n/a |
University of California at San Diego Curated by ChEMBL | Assay Description In vitro inhibition of radioligand binding to human somatostatin receptor (hsst3) expressed in CHO cells. | J Med Chem 41: 2679-85 (1998) Article DOI: 10.1021/jm970393l BindingDB Entry DOI: 10.7270/Q2Z60N6X | |||||||||||
More data for this Ligand-Target Pair |