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Compile Data Set for Download or QSAR

Found 1 hit Enz. Inhib. hit(s) with Target = 'Somatostatin receptor type 4' and Ligand = 'BDBM50136807'   
Target/Host
(Institution)		LigandTarget/Host
Links		Ligand
Links		Trg + Lig
Links		Ki
nM		ΔG°
kJ/mole		IC50
nM		Kd
nM		EC50/IC50
nM		koff
s-1		kon
M-1s-1		pHTemp
°C
Somatostatin receptor type 4


(Homo sapiens (Human))		BDBM50136807
PNG
(CHEMBL405735 | Somatostatin analogue)
Show SMILES C[C@@H](O)[C@H]1NC(=O)[C@H](CCCCN)NC(=O)[C@@H](Cc2c[nH]c3ccccc23)NC(=O)[C@H](Cc2ccc(N)cc2)NC(=O)[C@@H](Cc2ccccc2)NC(=O)[C@H](N)CSSC[C@H](NC(=O)[C@H](Cc2ccc(O)cc2)NC1=O)C(O)=O
Show InChI InChI=1S/C54H67N11O11S2/c1-30(66)46-53(74)63-43(25-33-16-20-36(67)21-17-33)51(72)64-45(54(75)76)29-78-77-28-38(57)47(68)60-41(23-31-9-3-2-4-10-31)49(70)61-42(24-32-14-18-35(56)19-15-32)50(71)62-44(26-34-27-58-39-12-6-5-11-37(34)39)52(73)59-40(48(69)65-46)13-7-8-22-55/h2-6,9-12,14-21,27,30,38,40-46,58,66-67H,7-8,13,22-26,28-29,55-57H2,1H3,(H,59,73)(H,60,68)(H,61,70)(H,62,71)(H,63,74)(H,64,72)(H,65,69)(H,75,76)/t30-,38-,40+,41-,42+,43+,44-,45+,46-/m1/s1
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Similars
Article
PubMed
n/an/a 1.10n/an/an/an/an/an/a



Salk Institute

Curated by ChEMBL


Assay Description
Binding affinity towards human somatostatin receptor type 4 using [125I]-[Leu8,DTrp22,Tyr25]SRIF-28 as radioligand.

J Med Chem 46: 5597-605 (2003)


Article DOI: 10.1021/jm030245x
BindingDB Entry DOI: 10.7270/Q2MK6C9X
More data for this
Ligand-Target Pair