Target/Host (Institution) | Ligand | Target/Host Links | Ligand Links | Trg + Lig Links | Ki nM | ΔG° kJ/mole | IC50 nM | Kd nM | EC50/IC50 nM | koff s-1 | kon M-1s-1 | pH | Temp °C |
---|---|---|---|---|---|---|---|---|---|---|---|---|---|
Sphingosine 1-phosphate receptor 1 (Homo sapiens (Human)) | BDBM50399042 (CHEMBL2178812) | PDB Reactome pathway KEGG UniProtKB/SwissProt B.MOAD antibodypedia GoogleScholar AffyNet | CHEMBL PC cid PC sid UniChem Similars | Article PubMed | n/a | n/a | 2.10 | n/a | n/a | n/a | n/a | n/a | n/a |
Novartis Pharma AG Curated by ChEMBL | Assay Description Antagonist activity at human S1P1R receptor expressed in CHO cell membranes by [35S]GTPgamma binding assay | J Med Chem 55: 9722-34 (2012) Article DOI: 10.1021/jm3009508 BindingDB Entry DOI: 10.7270/Q2K938PD | |||||||||||
More data for this Ligand-Target Pair |