Target/Host (Institution) | Ligand | Target/Host Links | Ligand Links | Trg + Lig Links | Ki nM | ΔG° kJ/mole | IC50 nM | Kd nM | EC50/IC50 nM | koff s-1 | kon M-1s-1 | pH | Temp °C |
---|---|---|---|---|---|---|---|---|---|---|---|---|---|
Sphingosine 1-phosphate receptor 3 (Homo sapiens (Human)) | BDBM50045325 (CHEMBL3311106) | PDB NCI pathway Reactome pathway KEGG UniProtKB/SwissProt antibodypedia GoogleScholar AffyNet | CHEMBL PC cid PC sid UniChem Patents Similars | Article PubMed | n/a | n/a | n/a | n/a | 200 | n/a | n/a | n/a | n/a |
Cardiff University Curated by ChEMBL | Assay Description Agonist activity at human S1P3 receptor expressed in CHOK1 cell membranes by [35S]-GTPgammaS binding assay | Bioorg Med Chem Lett 27: 1371-1378 (2017) Article DOI: 10.1016/j.bmcl.2017.02.011 BindingDB Entry DOI: 10.7270/Q27P91N1 | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Sphingosine 1-phosphate receptor 3 (Homo sapiens (Human)) | BDBM50045325 (CHEMBL3311106) | PDB NCI pathway Reactome pathway KEGG UniProtKB/SwissProt antibodypedia GoogleScholar AffyNet | CHEMBL PC cid PC sid UniChem Patents Similars | Article PubMed | n/a | n/a | n/a | n/a | 200 | n/a | n/a | n/a | n/a |
Daiichi Sankyo Co, Ltd Curated by ChEMBL | Assay Description Agonist activity at human S1P3 receptor expressed in CHOK1 cell membranes by [35S]GTPgammaS binding assay | Bioorg Med Chem 22: 4246-56 (2014) Article DOI: 10.1016/j.bmc.2014.05.035 BindingDB Entry DOI: 10.7270/Q2PN9788 | |||||||||||
More data for this Ligand-Target Pair |