Target/Host (Institution) | Ligand | Target/Host Links | Ligand Links | Trg + Lig Links | Ki nM | ΔG° kJ/mole | IC50 nM | Kd nM | EC50/IC50 nM | koff s-1 | kon M-1s-1 | pH | Temp °C |
---|---|---|---|---|---|---|---|---|---|---|---|---|---|
Sphingosine 1-phosphate receptor 5 (Homo sapiens (Human)) | BDBM149705 (US8975409, Example 9(3)) | PDB NCI pathway Reactome pathway KEGG UniProtKB/SwissProt DrugBank antibodypedia GoogleScholar AffyNet | PC cid PC sid UniChem | Article PubMed | n/a | n/a | >1.00E+4 | n/a | n/a | n/a | n/a | n/a | n/a |
Ono Pharmaceutical Co. Curated by ChEMBL | Assay Description Displacement of [33P]S1P from human S1P5 expressed in CHO-K1 cells by scintillation counter | Bioorg Med Chem Lett 25: 4387-92 (2015) Article DOI: 10.1016/j.bmcl.2015.09.022 BindingDB Entry DOI: 10.7270/Q2SX6G1K | |||||||||||
More data for this Ligand-Target Pair |