Target/Host (Institution) | Ligand | Target/Host Links | Ligand Links | Trg + Lig Links | Ki nM | ΔG° kJ/mole | IC50 nM | Kd nM | EC50/IC50 nM | koff s-1 | kon M-1s-1 | pH | Temp °C |
---|---|---|---|---|---|---|---|---|---|---|---|---|---|
Telomerase reverse transcriptase (Homo sapiens (Human)) | BDBM50412201 (CRYPTOLEPINE HYDROCHLORIDE | Cryptolepine) | PDB NCI pathway Reactome pathway KEGG UniProtKB/SwissProt DrugBank antibodypedia GoogleScholar AffyNet | KEGG PC cid PC sid PDB UniChem Similars | Article PubMed | n/a | n/a | 9.40E+3 | n/a | n/a | n/a | n/a | n/a | n/a |
Universit£ degli Studi"Magna Gr£cia" Curated by ChEMBL | Assay Description Inhibition of telomerase (unknown origin) by TRAP assay | Eur J Med Chem 68: 139-49 (2013) Article DOI: 10.1016/j.ejmech.2013.07.022 BindingDB Entry DOI: 10.7270/Q24J0GJB | |||||||||||
More data for this Ligand-Target Pair |