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Compile Data Set for Download or QSAR

Found 1 hit Enz. Inhib. hit(s) with Target = 'Translocator protein' and Ligand = 'BDBM279580'   
Target/Host
(Institution)		LigandTarget/Host
Links		Ligand
Links		Trg + Lig
Links		Ki
nM		ΔG°
kJ/mole		IC50
nM		Kd
nM		EC50/IC50
nM		koff
s-1		kon
M-1s-1		pHTemp
°C
Translocator protein


(Homo sapiens (Human))		BDBM279580
PNG
(US10035780, Compound 4)
Show SMILES CCN(CC)C(=O)Oc1nc(nc2ccccc12)-c1ccc(Br)cc1
Show InChI InChI=1S/C19H18BrN3O2/c1-3-23(4-2)19(24)25-18-15-7-5-6-8-16(15)21-17(22-18)13-9-11-14(20)12-10-13/h5-12H,3-4H2,1-2H3
KEGG

UniProtKB/SwissProt

DrugBank
antibodypedia
GoogleScholar
AffyNet 
PC cid
PC sid
UniChem
US Patent
 45n/an/an/an/an/an/an/an/a



TECHNION RESEARCH & DEVELOPMENT FOUNDATION LTD.

US Patent


Assay Description
For the assays described herein systemic injections of kainic in rats were applied and also contusion (Veenman et al. 2002; Soustiel et al. Neuropath...

US Patent US10035780 (2018)


BindingDB Entry DOI: 10.7270/Q20V8FTD
More data for this
Ligand-Target Pair