Target/Host (Institution) | Ligand | Target/Host Links | Ligand Links | Trg + Lig Links | Ki nM | ΔG° kJ/mole | IC50 nM | Kd nM | EC50/IC50 nM | koff s-1 | kon M-1s-1 | pH | Temp °C |
---|---|---|---|---|---|---|---|---|---|---|---|---|---|
Trypanothione reductase (Trypanosoma cruzi) | BDBM50352509 (CHEMBL1824848) | PDB MMDB KEGG UniProtKB/SwissProt B.MOAD DrugBank GoogleScholar AffyNet | CHEMBL PC cid PC sid UniChem | Article PubMed | 5.70E+3 | n/a | n/a | n/a | n/a | n/a | n/a | n/a | n/a |
Universit£ degli Studi di Siena Curated by ChEMBL | Assay Description Inhibition of Trypanosoma cruzi TryR using trypanothione as substrate preincubated for 10 mins | Bioorg Med Chem Lett 21: 5255-8 (2011) Article DOI: 10.1016/j.bmcl.2011.07.036 BindingDB Entry DOI: 10.7270/Q2ZP46HX | |||||||||||
More data for this Ligand-Target Pair |