Target/Host (Institution) | Ligand | Target/Host Links | Ligand Links | Trg + Lig Links | Ki nM | ΔG° kJ/mole | IC50 nM | Kd nM | EC50/IC50 nM | koff s-1 | kon M-1s-1 | pH | Temp °C |
---|---|---|---|---|---|---|---|---|---|---|---|---|---|
Tyrosine-protein kinase ABL1 (Homo sapiens (Human)) | BDBM50324796 (3-[1-(4-chlorobenzyl)-1H-indol-3-yl]-N-(4-nitrophe...) | PDB MMDB Reactome pathway KEGG UniProtKB/SwissProt B.MOAD DrugBank antibodypedia GoogleScholar AffyNet | CHEMBL KEGG PC cid PC sid UniChem Similars | Article PubMed | n/a | n/a | >1.00E+5 | n/a | n/a | n/a | n/a | n/a | n/a |
Université de Nantes Curated by ChEMBL | Assay Description Inhibition of recombinant c-Abl after 1 hr | Bioorg Med Chem Lett 20: 5203-6 (2010) Article DOI: 10.1016/j.bmcl.2010.07.001 BindingDB Entry DOI: 10.7270/Q21C1X3M | |||||||||||
More data for this Ligand-Target Pair |