Target/Host (Institution) | Ligand | Target/Host Links | Ligand Links | Trg + Lig Links | Ki nM | ΔG° kJ/mole | IC50 nM | Kd nM | EC50/IC50 nM | koff s-1 | kon M-1s-1 | pH | Temp °C |
---|---|---|---|---|---|---|---|---|---|---|---|---|---|
Tyrosine-protein kinase Lck (Homo sapiens (Human)) | BDBM50092231 ((4-Phenoxy-phenyl)-quinazolin-4-yl-amine | CHEMBL3...) | PDB UniProtKB/SwissProt antibodypedia GoogleScholar AffyNet | Purchase CHEMBL PC cid PC sid UniChem Patents Similars | PubMed | n/a | n/a | <8 | n/a | n/a | n/a | n/a | n/a | n/a |
BASF Bioresearch Corporation Curated by ChEMBL | Assay Description Inhibition of p56 Lck tyrosine kinase at 1 mM ATP | Bioorg Med Chem Lett 10: 2167-70 (2001) BindingDB Entry DOI: 10.7270/Q2J38RTH | |||||||||||
More data for this Ligand-Target Pair |