Target/Host (Institution) | Ligand | Target/Host Links | Ligand Links | Trg + Lig Links | Ki nM | ΔG° kJ/mole | IC50 nM | Kd nM | EC50/IC50 nM | koff s-1 | kon M-1s-1 | pH | Temp °C |
---|---|---|---|---|---|---|---|---|---|---|---|---|---|
Tyrosine-protein kinase Lck (Homo sapiens (Human)) | BDBM50114585 ((R)-7-[4-(4-Methyl-piperazin-1-yl)-cyclohexyl]-5-(...) | PDB UniProtKB/SwissProt antibodypedia GoogleScholar AffyNet | Purchase CHEMBL MMDB PC cid PC sid PDB UniChem Patents Similars | PubMed | n/a | n/a | 15 | n/a | n/a | n/a | n/a | n/a | n/a |
Abbott Bioresearch Center Curated by ChEMBL | Assay Description Inhibition of human p56 Lck tyrosine kinase (lck64-509) | Bioorg Med Chem Lett 12: 1683-6 (2002) BindingDB Entry DOI: 10.7270/Q23B5ZGR | |||||||||||
More data for this Ligand-Target Pair |