Target/Host (Institution) | Ligand | Target/Host Links | Ligand Links | Trg + Lig Links | Ki nM | ΔG° kJ/mole | IC50 nM | Kd nM | EC50/IC50 nM | koff s-1 | kon M-1s-1 | pH | Temp °C |
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Vasopressin V1a receptor (Homo sapiens (Human)) | BDBM50239342 (CHEMBL4075127) | PDB UniProtKB/SwissProt antibodypedia GoogleScholar AffyNet | CHEMBL PC cid PC sid UniChem | Article PubMed | 1 | n/a | n/a | n/a | n/a | n/a | n/a | n/a | n/a |
Teikyo University Curated by ChEMBL | Assay Description Displacement of [125I] phenylacetyl-D-Tyr(Me)-Phe-Gln-Asn-Arg-Pro-Arg-Tyr-NH2 from human recombinant vasopressin V1a receptor expressed in HEK293 aft... | J Med Chem 60: 4503-4509 (2017) Article DOI: 10.1021/acs.jmedchem.7b00422 BindingDB Entry DOI: 10.7270/Q27946TN | |||||||||||
More data for this Ligand-Target Pair |