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Compile Data Set for Download or QSAR

Found 1 hit Enz. Inhib. hit(s) with Target = 'Voltage-gated potassium channel' and Ligand = 'BDBM50278973'   
Target/Host
(Institution)
LigandTarget/Host
Links
Ligand
Links
Trg + Lig
Links
Ki
nM
ΔG°
kJ/mole
IC50
nM
Kd
nM
EC50/IC50
nM
koff
s-1
kon
M-1s-1
pHTemp
°C
Voltage-gated potassium channel


(Homo sapiens (Human))
BDBM50278973
PNG
((5-(furan-2-carbonyl)-5,6-dihydrophenanthridin-6-y...)
Show SMILES COc1ccccc1C(=O)C1N(C(=O)c2ccco2)c2ccccc2-c2ccccc12
Show InChI InChI=1S/C26H19NO4/c1-30-22-14-7-5-12-20(22)25(28)24-19-11-3-2-9-17(19)18-10-4-6-13-21(18)27(24)26(29)23-15-8-16-31-23/h2-16,24H,1H3
PDB
MMDB

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PC cid
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Article
PubMed
n/an/a 1.50E+3n/an/an/an/an/an/a



4SC AG

Curated by ChEMBL


Assay Description
Inhibition of cloned Kv1.3 channel (unknown origin) expressed in mammalian cells by whole cell patch clamp assay


Bioorg Med Chem Lett 19: 2299-304 (2009)


Article DOI: 10.1016/j.bmcl.2009.02.077
BindingDB Entry DOI: 10.7270/Q29K4B38
More data for this
Ligand-Target Pair