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Found 1 hit Enz. Inhib. hit(s) with Target = 'cAMP and cAMP-inhibited cGMP 3',5'-cyclic phosphodiesterase 10A' and Ligand = 'BDBM304037'   
Target/Host
(Institution)		LigandTarget/Host
Links		Ligand
Links		Trg + Lig
Links		Ki
nM		ΔG°
kJ/mole		IC50
nM		Kd
nM		EC50/IC50
nM		koff
s-1		kon
M-1s-1		pHTemp
°C
cAMP and cAMP-inhibited cGMP 3',5'-cyclic phosphodiesterase 10A


(Homo sapiens (Human))		BDBM304037
PNG
(5,8-Dimethyl-2-[2-(1,3-thiazol-2-yl)-1H-benz-imida...)
Show SMILES Cc1cnc(C)c2nc(nn12)-c1ccc2[nH]c(nc2c1)-c1nccs1
Show InChI InChI=1S/C17H13N7S/c1-9-8-19-10(2)16-22-14(23-24(9)16)11-3-4-12-13(7-11)21-15(20-12)17-18-5-6-25-17/h3-8H,1-2H3,(H,20,21)
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US Patent
n/an/a 84n/an/an/an/an/an/a



CELON PHARMA S.A.

US Patent


Assay Description
Recombinant human phosphodiesterase 10A (PDE10A) purified to homogeneity from Sf9 cells overexpressing PDE10A gene (GenBank/EMBL accession number: NM...

US Patent US10138245 (2018)


BindingDB Entry DOI: 10.7270/Q2M32XTX
More data for this
Ligand-Target Pair