Target/Host (Institution) | Ligand | Target/Host Links | Ligand Links | Trg + Lig Links | Ki nM | ΔG° kJ/mole | IC50 nM | Kd nM | EC50/IC50 nM | koff s-1 | kon M-1s-1 | pH | Temp °C |
---|---|---|---|---|---|---|---|---|---|---|---|---|---|
cAMP-specific 3',5'-cyclic phosphodiesterase 4B (Homo sapiens (Human)) | BDBM50363907 (CHEMBL1946748) | PDB UniProtKB/SwissProt antibodypedia GoogleScholar AffyNet | CHEMBL PC cid PC sid UniChem Patents | Article PubMed | n/a | n/a | 1.01E+3 | n/a | n/a | n/a | n/a | n/a | n/a |
Kyorin Pharmaceutical Co. Ltd. Curated by ChEMBL | Assay Description Inhibition of human PDE4B catalytic domain | Bioorg Med Chem 20: 1644-58 (2012) Article DOI: 10.1016/j.bmc.2012.01.033 BindingDB Entry DOI: 10.7270/Q2DB829P | |||||||||||
More data for this Ligand-Target Pair |