Target/Host (Institution) | Ligand | Target/Host Links | Ligand Links | Trg + Lig Links | Ki nM | ΔG° kJ/mole | IC50 nM | Kd nM | EC50/IC50 nM | koff s-1 | kon M-1s-1 | pH | Temp °C |
---|---|---|---|---|---|---|---|---|---|---|---|---|---|
histone lysine demethylase PHF8 isoform 2 (Homo sapiens (Human)) | BDBM276089![]() (1-(3-chlorophenyl)-4-{1H-[1,2,3]triazolo[4,5-c]pyr...) | PDB GoogleScholar AffyNet ![]() | PC cid PC sid UniChem | US Patent | n/a | n/a | 5.50E+3 | n/a | n/a | n/a | n/a | n/a | 25 |
Celgene Quanticel Research, Inc. US Patent | US Patent US10071984 (2018) BindingDB Entry DOI: 10.7270/Q24Q7X0X | ||||||||||||
More data for this Ligand-Target Pair |