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Compile Data Set for Download or QSAR

Found 82 hits with Last Name = 'blazer' and Initial = 'll'   
Target/Host
(Institution)
LigandTarget/Host
Links
Ligand
Links
Trg + Lig
Links
Ki
nM
ΔG°
kJ/mole
IC50
nM
Kd
nM
EC50/IC50
nM
koff
s-1
kon
M-1s-1
pHTemp
°C
Regulator of G-protein signaling 4 (RGS4)


(Homo sapiens (Human))
BDBM50384752
PNG
(CHEMBL2037351)
Show SMILES Cc1ccc(cc1)-n1sc(=O)n(Cc2ccc(Cl)cc2)c1=O
Show InChI InChI=1S/C16H13ClN2O2S/c1-11-2-8-14(9-3-11)19-15(20)18(16(21)22-19)10-12-4-6-13(17)7-5-12/h2-9H,10H2,1H3
PDB

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n/an/a 5.40n/an/an/an/an/an/a



TBA

Curated by ChEMBL


Assay Description
Inhibition of RGS4 interaction with Galpha0 protein by flow cytometry protein interaction assay


ACS Med Chem Lett 3: 146-150 (2012)


Article DOI: 10.1021/ml200263y
BindingDB Entry DOI: 10.7270/Q2NS0VXW
More data for this
Ligand-Target Pair
Regulator of G-protein signaling 4 (RGS4)


(Homo sapiens (Human))
BDBM50384751
PNG
(CHEMBL2037350)
Show SMILES Cc1ccc(Cn2sc(=O)n(Cc3ccccc3)c2=O)cc1
Show InChI InChI=1S/C17H16N2O2S/c1-13-7-9-15(10-8-13)12-19-16(20)18(17(21)22-19)11-14-5-3-2-4-6-14/h2-10H,11-12H2,1H3
PDB

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n/an/a 7.20n/an/an/an/an/an/a



TBA

Curated by ChEMBL


Assay Description
Inhibition of RGS4 interaction with Galpha0 protein by flow cytometry protein interaction assay


ACS Med Chem Lett 3: 146-150 (2012)


Article DOI: 10.1021/ml200263y
BindingDB Entry DOI: 10.7270/Q2NS0VXW
More data for this
Ligand-Target Pair
Regulator of G-protein signaling 4 (RGS4)


(Homo sapiens (Human))
BDBM50384755
PNG
(CHEMBL2037352)
Show SMILES Cc1ccc(Cn2c(=O)sn(-c3ccc(C)cc3)c2=O)cc1
Show InChI InChI=1S/C17H16N2O2S/c1-12-3-7-14(8-4-12)11-18-16(20)19(22-17(18)21)15-9-5-13(2)6-10-15/h3-10H,11H2,1-2H3
PDB

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n/an/a 8.60n/an/an/an/an/an/a



TBA

Curated by ChEMBL


Assay Description
Inhibition of RGS4 interaction with Galpha0 protein by flow cytometry protein interaction assay


ACS Med Chem Lett 3: 146-150 (2012)


Article DOI: 10.1021/ml200263y
BindingDB Entry DOI: 10.7270/Q2NS0VXW
More data for this
Ligand-Target Pair
Regulator of G-protein signaling 4 (RGS4)


(Homo sapiens (Human))
BDBM50384777
PNG
(CHEMBL2037229)
Show SMILES COc1ccc(cc1)-n1sc(=O)n(Cc2ccc(F)cc2)c1=O
Show InChI InChI=1S/C16H13FN2O3S/c1-22-14-8-6-13(7-9-14)19-15(20)18(16(21)23-19)10-11-2-4-12(17)5-3-11/h2-9H,10H2,1H3
PDB

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TBA

Curated by ChEMBL


Assay Description
Inhibition of RGS4 interaction with Galpha0 protein by flow cytometry protein interaction assay


ACS Med Chem Lett 3: 146-150 (2012)


Article DOI: 10.1021/ml200263y
BindingDB Entry DOI: 10.7270/Q2NS0VXW
More data for this
Ligand-Target Pair
Regulator of G-protein signaling 4 (RGS4)


(Homo sapiens (Human))
BDBM50384754
PNG
(CHEMBL2037234)
Show SMILES Cc1ccc(Cn2sc(=O)n(Cc3ccc(F)cc3)c2=O)cc1
Show InChI InChI=1S/C17H15FN2O2S/c1-12-2-4-14(5-3-12)11-20-16(21)19(17(22)23-20)10-13-6-8-15(18)9-7-13/h2-9H,10-11H2,1H3
PDB

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n/an/a 13n/an/an/an/an/an/a



TBA

Curated by ChEMBL


Assay Description
Inhibition of RGS4 interaction with Galpha0 protein by flow cytometry protein interaction assay


ACS Med Chem Lett 3: 146-150 (2012)


Article DOI: 10.1021/ml200263y
BindingDB Entry DOI: 10.7270/Q2NS0VXW
More data for this
Ligand-Target Pair
Regulator of G-protein signaling 4 (RGS4)


(Homo sapiens (Human))
BDBM50384776
PNG
(CHEMBL2037228)
Show SMILES Fc1ccc(Cn2c(=O)sn(-c3ccc(Cl)cc3)c2=O)cc1
Show InChI InChI=1S/C15H10ClFN2O2S/c16-11-3-7-13(8-4-11)19-14(20)18(15(21)22-19)9-10-1-5-12(17)6-2-10/h1-8H,9H2
PDB

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n/an/a 14n/an/an/an/an/an/a



TBA

Curated by ChEMBL


Assay Description
Inhibition of RGS4 interaction with Galpha0 protein by flow cytometry protein interaction assay


ACS Med Chem Lett 3: 146-150 (2012)


Article DOI: 10.1021/ml200263y
BindingDB Entry DOI: 10.7270/Q2NS0VXW
More data for this
Ligand-Target Pair
Regulator of G-protein signaling 4 (RGS4)


(Homo sapiens (Human))
BDBM50384743
PNG
(CHEMBL2037235)
Show SMILES Cc1ccc(cc1)-n1sc(=O)n(Cc2ccccc2)c1=O
Show InChI InChI=1S/C16H14N2O2S/c1-12-7-9-14(10-8-12)18-15(19)17(16(20)21-18)11-13-5-3-2-4-6-13/h2-10H,11H2,1H3
PDB

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TBA

Curated by ChEMBL


Assay Description
Inhibition of RGS4 interaction with Galpha0 protein by flow cytometry protein interaction assay


ACS Med Chem Lett 3: 146-150 (2012)


Article DOI: 10.1021/ml200263y
BindingDB Entry DOI: 10.7270/Q2NS0VXW
More data for this
Ligand-Target Pair
Regulator of G-protein signaling 4 (RGS4)


(Homo sapiens (Human))
BDBM7779
PNG
(4-butyl-2-ethyl-1,2,4-thiadiazolidine-3,5-dione | ...)
Show SMILES CCCCn1c(=O)sn(CC)c1=O
Show InChI InChI=1S/C8H14N2O2S/c1-3-5-6-9-7(11)10(4-2)13-8(9)12/h3-6H2,1-2H3
PDB

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n/an/a 14n/an/an/an/an/an/a



TBA

Curated by ChEMBL


Assay Description
Inhibition of RGS4 interaction with Galpha0 protein by flow cytometry protein interaction assay


ACS Med Chem Lett 3: 146-150 (2012)


Article DOI: 10.1021/ml200263y
BindingDB Entry DOI: 10.7270/Q2NS0VXW
More data for this
Ligand-Target Pair
Regulator of G-protein signaling 4 (RGS4)


(Homo sapiens (Human))
BDBM50384767
PNG
(CHEMBL2037365)
Show SMILES CC(C)Cn1c(=O)sn(-c2ccc(C)cc2)c1=O
Show InChI InChI=1S/C13H16N2O2S/c1-9(2)8-14-12(16)15(18-13(14)17)11-6-4-10(3)5-7-11/h4-7,9H,8H2,1-3H3
PDB

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TBA

Curated by ChEMBL


Assay Description
Inhibition of RGS4 interaction with Galpha0 protein by flow cytometry protein interaction assay


ACS Med Chem Lett 3: 146-150 (2012)


Article DOI: 10.1021/ml200263y
BindingDB Entry DOI: 10.7270/Q2NS0VXW
More data for this
Ligand-Target Pair
Regulator of G-protein signaling 4 (RGS4)


(Homo sapiens (Human))
BDBM50384757
PNG
(CHEMBL2037354)
Show SMILES Cc1ccc(cc1)-n1sc(=O)n(Cc2cccc(C)c2)c1=O
Show InChI InChI=1S/C17H16N2O2S/c1-12-6-8-15(9-7-12)19-16(20)18(17(21)22-19)11-14-5-3-4-13(2)10-14/h3-10H,11H2,1-2H3
PDB

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n/an/a 15n/an/an/an/an/an/a



TBA

Curated by ChEMBL


Assay Description
Inhibition of RGS4 interaction with Galpha0 protein by flow cytometry protein interaction assay


ACS Med Chem Lett 3: 146-150 (2012)


Article DOI: 10.1021/ml200263y
BindingDB Entry DOI: 10.7270/Q2NS0VXW
More data for this
Ligand-Target Pair
Regulator of G-protein signaling 4 (RGS4)


(Homo sapiens (Human))
BDBM50384775
PNG
(CHEMBL2037227)
Show SMILES Fc1ccc(Cn2c(=O)sn(-c3ccccc3)c2=O)cc1
Show InChI InChI=1S/C15H11FN2O2S/c16-12-8-6-11(7-9-12)10-17-14(19)18(21-15(17)20)13-4-2-1-3-5-13/h1-9H,10H2
PDB

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n/an/a 16n/an/an/an/an/an/a



TBA

Curated by ChEMBL


Assay Description
Inhibition of RGS4 interaction with Galpha0 protein by flow cytometry protein interaction assay


ACS Med Chem Lett 3: 146-150 (2012)


Article DOI: 10.1021/ml200263y
BindingDB Entry DOI: 10.7270/Q2NS0VXW
More data for this
Ligand-Target Pair
Regulator of G-protein signaling 4 (RGS4)


(Homo sapiens (Human))
BDBM50384760
PNG
(CHEMBL2035006)
Show SMILES CCCCn1sc(=O)n(Cc2ccc(F)cc2)c1=O
Show InChI InChI=1S/C13H15FN2O2S/c1-2-3-8-16-12(17)15(13(18)19-16)9-10-4-6-11(14)7-5-10/h4-7H,2-3,8-9H2,1H3
PDB

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n/an/a 16n/an/an/an/an/an/a



TBA

Curated by ChEMBL


Assay Description
Inhibition of RGS4 interaction with Galpha0 protein by flow cytometry protein interaction assay


ACS Med Chem Lett 3: 146-150 (2012)


Article DOI: 10.1021/ml200263y
BindingDB Entry DOI: 10.7270/Q2NS0VXW
More data for this
Ligand-Target Pair
Regulator of G-protein signaling 4 (RGS4)


(Homo sapiens (Human))
BDBM50384756
PNG
(CHEMBL2037353)
Show SMILES Cc1ccc(cc1)-n1sc(=O)n(Cc2cccc(Cl)c2)c1=O
Show InChI InChI=1S/C16H13ClN2O2S/c1-11-5-7-14(8-6-11)19-15(20)18(16(21)22-19)10-12-3-2-4-13(17)9-12/h2-9H,10H2,1H3
PDB

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n/an/a 17n/an/an/an/an/an/a



TBA

Curated by ChEMBL


Assay Description
Inhibition of RGS4 interaction with Galpha0 protein by flow cytometry protein interaction assay


ACS Med Chem Lett 3: 146-150 (2012)


Article DOI: 10.1021/ml200263y
BindingDB Entry DOI: 10.7270/Q2NS0VXW
More data for this
Ligand-Target Pair
Regulator of G-protein signaling 4 (RGS4)


(Homo sapiens (Human))
BDBM50384761
PNG
(CHEMBL2037358)
Show SMILES Cc1ccc(cc1)-n1sc(=O)n(C)c1=O
Show InChI InChI=1S/C10H10N2O2S/c1-7-3-5-8(6-4-7)12-9(13)11(2)10(14)15-12/h3-6H,1-2H3
PDB

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n/an/a 19n/an/an/an/an/an/a



TBA

Curated by ChEMBL


Assay Description
Inhibition of RGS4 interaction with Galpha0 protein by flow cytometry protein interaction assay


ACS Med Chem Lett 3: 146-150 (2012)


Article DOI: 10.1021/ml200263y
BindingDB Entry DOI: 10.7270/Q2NS0VXW
More data for this
Ligand-Target Pair
Regulator of G-protein signaling 4 (RGS4)


(Homo sapiens (Human))
BDBM50384764
PNG
(CHEMBL2037362)
Show SMILES CCCCn1c(=O)sn(-c2ccc(C)cc2)c1=O
Show InChI InChI=1S/C13H16N2O2S/c1-3-4-9-14-12(16)15(18-13(14)17)11-7-5-10(2)6-8-11/h5-8H,3-4,9H2,1-2H3
PDB

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n/an/a 20n/an/an/an/an/an/a



TBA

Curated by ChEMBL


Assay Description
Inhibition of RGS4 interaction with Galpha0 protein by flow cytometry protein interaction assay


ACS Med Chem Lett 3: 146-150 (2012)


Article DOI: 10.1021/ml200263y
BindingDB Entry DOI: 10.7270/Q2NS0VXW
More data for this
Ligand-Target Pair
Regulator of G-protein signaling 4 (RGS4)


(Homo sapiens (Human))
BDBM50384762
PNG
(CHEMBL2037359)
Show SMILES CCn1sc(=O)n(C)c1=O
Show InChI InChI=1S/C5H8N2O2S/c1-3-7-4(8)6(2)5(9)10-7/h3H2,1-2H3
PDB

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n/an/a 22n/an/an/an/an/an/a



TBA

Curated by ChEMBL


Assay Description
Inhibition of RGS4 interaction with Galpha0 protein by flow cytometry protein interaction assay


ACS Med Chem Lett 3: 146-150 (2012)


Article DOI: 10.1021/ml200263y
BindingDB Entry DOI: 10.7270/Q2NS0VXW
More data for this
Ligand-Target Pair
Regulator of G-protein signaling 4 (RGS4)


(Homo sapiens (Human))
BDBM50384739
PNG
(CHEMBL2037357)
Show SMILES CCn1sc(=O)n(Cc2ccc(F)cc2)c1=O
Show InChI InChI=1S/C11H11FN2O2S/c1-2-14-10(15)13(11(16)17-14)7-8-3-5-9(12)6-4-8/h3-6H,2,7H2,1H3
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n/an/a 22n/an/an/an/an/an/a



TBA

Curated by ChEMBL


Assay Description
Inhibition of RGS4 interaction with Galpha0 protein by flow cytometry protein interaction assay


ACS Med Chem Lett 3: 146-150 (2012)


Article DOI: 10.1021/ml200263y
BindingDB Entry DOI: 10.7270/Q2NS0VXW
More data for this
Ligand-Target Pair
Regulator of G-protein signaling 4 (RGS4)


(Homo sapiens (Human))
BDBM50384744
PNG
(CHEMBL2037236)
Show SMILES O=c1sn(-c2ccccc2)c(=O)n1Cc1ccccc1
Show InChI InChI=1S/C15H12N2O2S/c18-14-16(11-12-7-3-1-4-8-12)15(19)20-17(14)13-9-5-2-6-10-13/h1-10H,11H2
PDB

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TBA

Curated by ChEMBL


Assay Description
Inhibition of RGS4 interaction with Galpha0 protein by flow cytometry protein interaction assay


ACS Med Chem Lett 3: 146-150 (2012)


Article DOI: 10.1021/ml200263y
BindingDB Entry DOI: 10.7270/Q2NS0VXW
More data for this
Ligand-Target Pair
Regulator of G-protein signaling 4 (RGS4)


(Homo sapiens (Human))
BDBM50384763
PNG
(CHEMBL2037360)
Show SMILES CCCCn1sc(=O)n(C)c1=O
Show InChI InChI=1S/C7H12N2O2S/c1-3-4-5-9-6(10)8(2)7(11)12-9/h3-5H2,1-2H3
PDB

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TBA

Curated by ChEMBL


Assay Description
Inhibition of RGS4 interaction with Galpha0 protein by flow cytometry protein interaction assay


ACS Med Chem Lett 3: 146-150 (2012)


Article DOI: 10.1021/ml200263y
BindingDB Entry DOI: 10.7270/Q2NS0VXW
More data for this
Ligand-Target Pair
Regulator of G-protein signaling 4 (RGS4)


(Homo sapiens (Human))
BDBM50384746
PNG
(CHEMBL2037238)
Show SMILES COc1ccc(cc1)-n1sc(=O)n(Cc2ccccc2)c1=O
Show InChI InChI=1S/C16H14N2O3S/c1-21-14-9-7-13(8-10-14)18-15(19)17(16(20)22-18)11-12-5-3-2-4-6-12/h2-10H,11H2,1H3
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TBA

Curated by ChEMBL


Assay Description
Inhibition of RGS4 interaction with Galpha0 protein by flow cytometry protein interaction assay


ACS Med Chem Lett 3: 146-150 (2012)


Article DOI: 10.1021/ml200263y
BindingDB Entry DOI: 10.7270/Q2NS0VXW
More data for this
Ligand-Target Pair
Regulator of G-protein signaling 4 (RGS4)


(Homo sapiens (Human))
BDBM50384768
PNG
(CHEMBL2037366)
Show SMILES CCn1sc(=O)n(CC(C)C)c1=O
Show InChI InChI=1S/C8H14N2O2S/c1-4-10-7(11)9(5-6(2)3)8(12)13-10/h6H,4-5H2,1-3H3
PDB

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n/an/a 26n/an/an/an/an/an/a



TBA

Curated by ChEMBL


Assay Description
Inhibition of RGS4 interaction with Galpha0 protein by flow cytometry protein interaction assay


ACS Med Chem Lett 3: 146-150 (2012)


Article DOI: 10.1021/ml200263y
BindingDB Entry DOI: 10.7270/Q2NS0VXW
More data for this
Ligand-Target Pair
Regulator of G-protein signaling 4 (RGS4)


(Homo sapiens (Human))
BDBM50384753
PNG
(CHEMBL2037361)
Show SMILES Cn1c(=O)sn(c1=O)C(C)(C)C
Show InChI InChI=1S/C7H12N2O2S/c1-7(2,3)9-5(10)8(4)6(11)12-9/h1-4H3
PDB

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n/an/a 28n/an/an/an/an/an/a



TBA

Curated by ChEMBL


Assay Description
Inhibition of RGS4 interaction with Galpha0 protein by flow cytometry protein interaction assay


ACS Med Chem Lett 3: 146-150 (2012)


Article DOI: 10.1021/ml200263y
BindingDB Entry DOI: 10.7270/Q2NS0VXW
More data for this
Ligand-Target Pair
Regulator of G-protein signaling 4 (RGS4)


(Homo sapiens (Human))
BDBM50384770
PNG
(CHEMBL2037368)
Show SMILES CC(C)Cn1c(=O)sn(c1=O)C(C)(C)C
Show InChI InChI=1S/C10H18N2O2S/c1-7(2)6-11-8(13)12(10(3,4)5)15-9(11)14/h7H,6H2,1-5H3
PDB

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TBA

Curated by ChEMBL


Assay Description
Inhibition of RGS4 interaction with Galpha0 protein by flow cytometry protein interaction assay


ACS Med Chem Lett 3: 146-150 (2012)


Article DOI: 10.1021/ml200263y
BindingDB Entry DOI: 10.7270/Q2NS0VXW
More data for this
Ligand-Target Pair
Regulator of G-protein signaling 4 (RGS4)


(Homo sapiens (Human))
BDBM50384745
PNG
(CHEMBL2037237)
Show SMILES Clc1ccc(cc1)-n1sc(=O)n(Cc2ccccc2)c1=O
Show InChI InChI=1S/C15H11ClN2O2S/c16-12-6-8-13(9-7-12)18-14(19)17(15(20)21-18)10-11-4-2-1-3-5-11/h1-9H,10H2
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TBA

Curated by ChEMBL


Assay Description
Inhibition of RGS4 interaction with Galpha0 protein by flow cytometry protein interaction assay


ACS Med Chem Lett 3: 146-150 (2012)


Article DOI: 10.1021/ml200263y
BindingDB Entry DOI: 10.7270/Q2NS0VXW
More data for this
Ligand-Target Pair
Regulator of G-protein signaling 4 (RGS4)


(Homo sapiens (Human))
BDBM50384774
PNG
(CHEMBL1917204)
Show SMILES Cc1ccc(cc1)-n1sc(=O)n(Cc2ccc(F)cc2)c1=O
Show InChI InChI=1S/C16H13FN2O2S/c1-11-2-8-14(9-3-11)19-15(20)18(16(21)22-19)10-12-4-6-13(17)7-5-12/h2-9H,10H2,1H3
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TBA

Curated by ChEMBL


Assay Description
Inhibition of RGS4 interaction with Galpha0 protein by flow cytometry protein interaction assay


ACS Med Chem Lett 3: 146-150 (2012)


Article DOI: 10.1021/ml200263y
BindingDB Entry DOI: 10.7270/Q2NS0VXW
More data for this
Ligand-Target Pair
Regulator of G-protein signaling 4 (RGS4)


(Homo sapiens (Human))
BDBM50384765
PNG
(CHEMBL2037363)
Show SMILES CCCCn1sc(=O)n(CCCC)c1=O
Show InChI InChI=1S/C10H18N2O2S/c1-3-5-7-11-9(13)12(8-6-4-2)15-10(11)14/h3-8H2,1-2H3
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TBA

Curated by ChEMBL


Assay Description
Inhibition of RGS4 interaction with Galpha0 protein by flow cytometry protein interaction assay


ACS Med Chem Lett 3: 146-150 (2012)


Article DOI: 10.1021/ml200263y
BindingDB Entry DOI: 10.7270/Q2NS0VXW
More data for this
Ligand-Target Pair
Regulator of G-protein signaling 4 (RGS4)


(Homo sapiens (Human))
BDBM50384750
PNG
(CHEMBL2037349)
Show SMILES Clc1cccc(c1)-n1sc(=O)n(Cc2ccccc2)c1=O
Show InChI InChI=1S/C15H11ClN2O2S/c16-12-7-4-8-13(9-12)18-14(19)17(15(20)21-18)10-11-5-2-1-3-6-11/h1-9H,10H2
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TBA

Curated by ChEMBL


Assay Description
Inhibition of RGS4 interaction with Galpha0 protein by flow cytometry protein interaction assay


ACS Med Chem Lett 3: 146-150 (2012)


Article DOI: 10.1021/ml200263y
BindingDB Entry DOI: 10.7270/Q2NS0VXW
More data for this
Ligand-Target Pair
Regulator of G-protein signaling 4 (RGS4)


(Homo sapiens (Human))
BDBM50384759
PNG
(CHEMBL2037356)
Show SMILES Cc1ccc(cc1)-n1sc(=O)n(Cc2ccc(Cl)c(Cl)c2)c1=O
Show InChI InChI=1S/C16H12Cl2N2O2S/c1-10-2-5-12(6-3-10)20-15(21)19(16(22)23-20)9-11-4-7-13(17)14(18)8-11/h2-8H,9H2,1H3
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TBA

Curated by ChEMBL


Assay Description
Inhibition of RGS4 interaction with Galpha0 protein by flow cytometry protein interaction assay


ACS Med Chem Lett 3: 146-150 (2012)


Article DOI: 10.1021/ml200263y
BindingDB Entry DOI: 10.7270/Q2NS0VXW
More data for this
Ligand-Target Pair
Regulator of G-protein signaling 4 (RGS4)


(Homo sapiens (Human))
BDBM50384778
PNG
(CHEMBL2037230)
Show SMILES Fc1ccc(Cn2c(=O)sn(-c3ccc(Cl)c(Cl)c3)c2=O)cc1
Show InChI InChI=1S/C15H9Cl2FN2O2S/c16-12-6-5-11(7-13(12)17)20-14(21)19(15(22)23-20)8-9-1-3-10(18)4-2-9/h1-7H,8H2
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TBA

Curated by ChEMBL


Assay Description
Inhibition of RGS4 interaction with Galpha0 protein by flow cytometry protein interaction assay


ACS Med Chem Lett 3: 146-150 (2012)


Article DOI: 10.1021/ml200263y
BindingDB Entry DOI: 10.7270/Q2NS0VXW
More data for this
Ligand-Target Pair
Regulator of G-protein signaling 4 (RGS4)


(Homo sapiens (Human))
BDBM50384749
PNG
(CHEMBL2037348)
Show SMILES Cc1cccc(c1)-n1sc(=O)n(Cc2ccccc2)c1=O
Show InChI InChI=1S/C16H14N2O2S/c1-12-6-5-9-14(10-12)18-15(19)17(16(20)21-18)11-13-7-3-2-4-8-13/h2-10H,11H2,1H3
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TBA

Curated by ChEMBL


Assay Description
Inhibition of RGS4 interaction with Galpha0 protein by flow cytometry protein interaction assay


ACS Med Chem Lett 3: 146-150 (2012)


Article DOI: 10.1021/ml200263y
BindingDB Entry DOI: 10.7270/Q2NS0VXW
More data for this
Ligand-Target Pair
Regulator of G-protein signaling 4 (RGS4)


(Homo sapiens (Human))
BDBM50384769
PNG
(CHEMBL2037367)
Show SMILES CCCCn1sc(=O)n(CC(C)C)c1=O
Show InChI InChI=1S/C10H18N2O2S/c1-4-5-6-12-9(13)11(7-8(2)3)10(14)15-12/h8H,4-7H2,1-3H3
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TBA

Curated by ChEMBL


Assay Description
Inhibition of RGS4 interaction with Galpha0 protein by flow cytometry protein interaction assay


ACS Med Chem Lett 3: 146-150 (2012)


Article DOI: 10.1021/ml200263y
BindingDB Entry DOI: 10.7270/Q2NS0VXW
More data for this
Ligand-Target Pair
Regulator of G-protein signaling 4 (RGS4)


(Homo sapiens (Human))
BDBM50384742
PNG
(CHEMBL2037233)
Show SMILES Fc1ccc(Cn2c(=O)sn(-c3cccc(Cl)c3)c2=O)cc1
Show InChI InChI=1S/C15H10ClFN2O2S/c16-11-2-1-3-13(8-11)19-14(20)18(15(21)22-19)9-10-4-6-12(17)7-5-10/h1-8H,9H2
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TBA

Curated by ChEMBL


Assay Description
Inhibition of RGS4 interaction with Galpha0 protein by flow cytometry protein interaction assay


ACS Med Chem Lett 3: 146-150 (2012)


Article DOI: 10.1021/ml200263y
BindingDB Entry DOI: 10.7270/Q2NS0VXW
More data for this
Ligand-Target Pair
Regulator of G-protein signaling 4 (RGS4)


(Homo sapiens (Human))
BDBM50384766
PNG
(CHEMBL2037364)
Show SMILES CCCCn1c(=O)sn(c1=O)C(C)(C)C
Show InChI InChI=1S/C10H18N2O2S/c1-5-6-7-11-8(13)12(10(2,3)4)15-9(11)14/h5-7H2,1-4H3
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TBA

Curated by ChEMBL


Assay Description
Inhibition of RGS4 interaction with Galpha0 protein by flow cytometry protein interaction assay


ACS Med Chem Lett 3: 146-150 (2012)


Article DOI: 10.1021/ml200263y
BindingDB Entry DOI: 10.7270/Q2NS0VXW
More data for this
Ligand-Target Pair
Regulator of G-protein signaling 4 (RGS4)


(Homo sapiens (Human))
BDBM50384771
PNG
(CHEMBL2037369)
Show SMILES CCn1sc(=O)n(CCOC)c1=O
Show InChI InChI=1S/C7H12N2O3S/c1-3-9-6(10)8(4-5-12-2)7(11)13-9/h3-5H2,1-2H3
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TBA

Curated by ChEMBL


Assay Description
Inhibition of RGS4 interaction with Galpha0 protein by flow cytometry protein interaction assay


ACS Med Chem Lett 3: 146-150 (2012)


Article DOI: 10.1021/ml200263y
BindingDB Entry DOI: 10.7270/Q2NS0VXW
More data for this
Ligand-Target Pair
Regulator of G-protein signaling 4 (RGS4)


(Homo sapiens (Human))
BDBM50384748
PNG
(CHEMBL2037347)
Show SMILES FC(F)(F)c1cccc(c1)-n1sc(=O)n(Cc2ccccc2)c1=O
Show InChI InChI=1S/C16H11F3N2O2S/c17-16(18,19)12-7-4-8-13(9-12)21-14(22)20(15(23)24-21)10-11-5-2-1-3-6-11/h1-9H,10H2
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TBA

Curated by ChEMBL


Assay Description
Inhibition of RGS4 interaction with Galpha0 protein by flow cytometry protein interaction assay


ACS Med Chem Lett 3: 146-150 (2012)


Article DOI: 10.1021/ml200263y
BindingDB Entry DOI: 10.7270/Q2NS0VXW
More data for this
Ligand-Target Pair
Regulator of G-protein signaling 4 (RGS4)


(Homo sapiens (Human))
BDBM50384740
PNG
(CHEMBL2037231)
Show SMILES Fc1ccc(Cn2c(=O)sn(-c3cccc(c3)C(F)(F)F)c2=O)cc1
Show InChI InChI=1S/C16H10F4N2O2S/c17-12-6-4-10(5-7-12)9-21-14(23)22(25-15(21)24)13-3-1-2-11(8-13)16(18,19)20/h1-8H,9H2
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TBA

Curated by ChEMBL


Assay Description
Inhibition of RGS4 interaction with Galpha0 protein by flow cytometry protein interaction assay


ACS Med Chem Lett 3: 146-150 (2012)


Article DOI: 10.1021/ml200263y
BindingDB Entry DOI: 10.7270/Q2NS0VXW
More data for this
Ligand-Target Pair
Regulator of G-protein signaling 4 (RGS4)


(Homo sapiens (Human))
BDBM50384747
PNG
(CHEMBL2037346)
Show SMILES Clc1ccc(cc1Cl)-n1sc(=O)n(Cc2ccccc2)c1=O
Show InChI InChI=1S/C15H10Cl2N2O2S/c16-12-7-6-11(8-13(12)17)19-14(20)18(15(21)22-19)9-10-4-2-1-3-5-10/h1-8H,9H2
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TBA

Curated by ChEMBL


Assay Description
Inhibition of RGS4 interaction with Galpha0 protein by flow cytometry protein interaction assay


ACS Med Chem Lett 3: 146-150 (2012)


Article DOI: 10.1021/ml200263y
BindingDB Entry DOI: 10.7270/Q2NS0VXW
More data for this
Ligand-Target Pair
Regulator of G-protein signaling 4 (RGS4)


(Homo sapiens (Human))
BDBM50384741
PNG
(CHEMBL2037232)
Show SMILES Cc1cccc(c1)-n1sc(=O)n(Cc2ccc(F)cc2)c1=O
Show InChI InChI=1S/C16H13FN2O2S/c1-11-3-2-4-14(9-11)19-15(20)18(16(21)22-19)10-12-5-7-13(17)8-6-12/h2-9H,10H2,1H3
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TBA

Curated by ChEMBL


Assay Description
Inhibition of RGS4 interaction with Galpha0 protein by flow cytometry protein interaction assay


ACS Med Chem Lett 3: 146-150 (2012)


Article DOI: 10.1021/ml200263y
BindingDB Entry DOI: 10.7270/Q2NS0VXW
More data for this
Ligand-Target Pair
Regulator of G-protein signaling 4 (RGS4)


(Homo sapiens (Human))
BDBM50384758
PNG
(CHEMBL2037355)
Show SMILES COc1ccc(Cn2c(=O)sn(-c3ccc(C)cc3)c2=O)cc1
Show InChI InChI=1S/C17H16N2O3S/c1-12-3-7-14(8-4-12)19-16(20)18(17(21)23-19)11-13-5-9-15(22-2)10-6-13/h3-10H,11H2,1-2H3
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TBA

Curated by ChEMBL


Assay Description
Inhibition of RGS4 interaction with Galpha0 protein by flow cytometry protein interaction assay


ACS Med Chem Lett 3: 146-150 (2012)


Article DOI: 10.1021/ml200263y
BindingDB Entry DOI: 10.7270/Q2NS0VXW
More data for this
Ligand-Target Pair
Regulator of G-protein signaling 8


(Homo sapiens (Human))
BDBM50384745
PNG
(CHEMBL2037237)
Show SMILES Clc1ccc(cc1)-n1sc(=O)n(Cc2ccccc2)c1=O
Show InChI InChI=1S/C15H11ClN2O2S/c16-12-6-8-13(9-7-12)18-14(19)17(15(20)21-18)10-11-4-2-1-3-5-11/h1-9H,10H2
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TBA

Curated by ChEMBL


Assay Description
Inhibition of RGS8 interaction with Galpha0 protein by flow cytometry protein interaction assay


ACS Med Chem Lett 3: 146-150 (2012)


Article DOI: 10.1021/ml200263y
BindingDB Entry DOI: 10.7270/Q2NS0VXW
More data for this
Ligand-Target Pair
Regulator of G-protein signaling 8


(Homo sapiens (Human))
BDBM50384744
PNG
(CHEMBL2037236)
Show SMILES O=c1sn(-c2ccccc2)c(=O)n1Cc1ccccc1
Show InChI InChI=1S/C15H12N2O2S/c18-14-16(11-12-7-3-1-4-8-12)15(19)20-17(14)13-9-5-2-6-10-13/h1-10H,11H2
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TBA

Curated by ChEMBL


Assay Description
Inhibition of RGS8 interaction with Galpha0 protein by flow cytometry protein interaction assay


ACS Med Chem Lett 3: 146-150 (2012)


Article DOI: 10.1021/ml200263y
BindingDB Entry DOI: 10.7270/Q2NS0VXW
More data for this
Ligand-Target Pair
Regulator of G-protein signaling 8


(Homo sapiens (Human))
BDBM50384775
PNG
(CHEMBL2037227)
Show SMILES Fc1ccc(Cn2c(=O)sn(-c3ccccc3)c2=O)cc1
Show InChI InChI=1S/C15H11FN2O2S/c16-12-8-6-11(7-9-12)10-17-14(19)18(21-15(17)20)13-4-2-1-3-5-13/h1-9H,10H2
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TBA

Curated by ChEMBL


Assay Description
Inhibition of RGS8 interaction with Galpha0 protein by flow cytometry protein interaction assay


ACS Med Chem Lett 3: 146-150 (2012)


Article DOI: 10.1021/ml200263y
BindingDB Entry DOI: 10.7270/Q2NS0VXW
More data for this
Ligand-Target Pair
Regulator of G-protein signaling 8


(Homo sapiens (Human))
BDBM50384741
PNG
(CHEMBL2037232)
Show SMILES Cc1cccc(c1)-n1sc(=O)n(Cc2ccc(F)cc2)c1=O
Show InChI InChI=1S/C16H13FN2O2S/c1-11-3-2-4-14(9-11)19-15(20)18(16(21)22-19)10-12-5-7-13(17)8-6-12/h2-9H,10H2,1H3
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TBA

Curated by ChEMBL


Assay Description
Inhibition of RGS8 interaction with Galpha0 protein by flow cytometry protein interaction assay


ACS Med Chem Lett 3: 146-150 (2012)


Article DOI: 10.1021/ml200263y
BindingDB Entry DOI: 10.7270/Q2NS0VXW
More data for this
Ligand-Target Pair
Regulator of G-protein signaling 8


(Homo sapiens (Human))
BDBM50384743
PNG
(CHEMBL2037235)
Show SMILES Cc1ccc(cc1)-n1sc(=O)n(Cc2ccccc2)c1=O
Show InChI InChI=1S/C16H14N2O2S/c1-12-7-9-14(10-8-12)18-15(19)17(16(20)21-18)11-13-5-3-2-4-6-13/h2-10H,11H2,1H3
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TBA

Curated by ChEMBL


Assay Description
Inhibition of RGS8 interaction with Galpha0 protein by flow cytometry protein interaction assay


ACS Med Chem Lett 3: 146-150 (2012)


Article DOI: 10.1021/ml200263y
BindingDB Entry DOI: 10.7270/Q2NS0VXW
More data for this
Ligand-Target Pair
Regulator of G-protein signaling 8


(Homo sapiens (Human))
BDBM50384776
PNG
(CHEMBL2037228)
Show SMILES Fc1ccc(Cn2c(=O)sn(-c3ccc(Cl)cc3)c2=O)cc1
Show InChI InChI=1S/C15H10ClFN2O2S/c16-11-3-7-13(8-4-11)19-14(20)18(15(21)22-19)9-10-1-5-12(17)6-2-10/h1-8H,9H2
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TBA

Curated by ChEMBL


Assay Description
Inhibition of RGS8 interaction with Galpha0 protein by flow cytometry protein interaction assay


ACS Med Chem Lett 3: 146-150 (2012)


Article DOI: 10.1021/ml200263y
BindingDB Entry DOI: 10.7270/Q2NS0VXW
More data for this
Ligand-Target Pair
Regulator of G-protein signaling 8


(Homo sapiens (Human))
BDBM50384767
PNG
(CHEMBL2037365)
Show SMILES CC(C)Cn1c(=O)sn(-c2ccc(C)cc2)c1=O
Show InChI InChI=1S/C13H16N2O2S/c1-9(2)8-14-12(16)15(18-13(14)17)11-6-4-10(3)5-7-11/h4-7,9H,8H2,1-3H3
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TBA

Curated by ChEMBL


Assay Description
Inhibition of RGS8 interaction with Galpha0 protein by flow cytometry protein interaction assay


ACS Med Chem Lett 3: 146-150 (2012)


Article DOI: 10.1021/ml200263y
BindingDB Entry DOI: 10.7270/Q2NS0VXW
More data for this
Ligand-Target Pair
Regulator of G-protein signaling 8


(Homo sapiens (Human))
BDBM50384761
PNG
(CHEMBL2037358)
Show SMILES Cc1ccc(cc1)-n1sc(=O)n(C)c1=O
Show InChI InChI=1S/C10H10N2O2S/c1-7-3-5-8(6-4-7)12-9(13)11(2)10(14)15-12/h3-6H,1-2H3
PDB
MMDB

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PC sid
UniChem
Article
PubMed
n/an/a 8.40E+3n/an/an/an/an/an/a



TBA

Curated by ChEMBL


Assay Description
Inhibition of RGS8 interaction with Galpha0 protein by flow cytometry protein interaction assay


ACS Med Chem Lett 3: 146-150 (2012)


Article DOI: 10.1021/ml200263y
BindingDB Entry DOI: 10.7270/Q2NS0VXW
More data for this
Ligand-Target Pair
Regulator of G-protein signaling 8


(Homo sapiens (Human))
BDBM50384764
PNG
(CHEMBL2037362)
Show SMILES CCCCn1c(=O)sn(-c2ccc(C)cc2)c1=O
Show InChI InChI=1S/C13H16N2O2S/c1-3-4-9-14-12(16)15(18-13(14)17)11-7-5-10(2)6-8-11/h5-8H,3-4,9H2,1-2H3
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n/an/a 9.50E+3n/an/an/an/an/an/a



TBA

Curated by ChEMBL


Assay Description
Inhibition of RGS8 interaction with Galpha0 protein by flow cytometry protein interaction assay


ACS Med Chem Lett 3: 146-150 (2012)


Article DOI: 10.1021/ml200263y
BindingDB Entry DOI: 10.7270/Q2NS0VXW
More data for this
Ligand-Target Pair
Regulator of G-protein signaling 8


(Homo sapiens (Human))
BDBM50384757
PNG
(CHEMBL2037354)
Show SMILES Cc1ccc(cc1)-n1sc(=O)n(Cc2cccc(C)c2)c1=O
Show InChI InChI=1S/C17H16N2O2S/c1-12-6-8-15(9-7-12)19-16(20)18(17(21)22-19)11-14-5-3-4-13(2)10-14/h3-10H,11H2,1-2H3
PDB
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n/an/a 9.90E+3n/an/an/an/an/an/a



TBA

Curated by ChEMBL


Assay Description
Inhibition of RGS8 interaction with Galpha0 protein by flow cytometry protein interaction assay


ACS Med Chem Lett 3: 146-150 (2012)


Article DOI: 10.1021/ml200263y
BindingDB Entry DOI: 10.7270/Q2NS0VXW
More data for this
Ligand-Target Pair
Regulator of G-protein signaling 8


(Homo sapiens (Human))
BDBM50384750
PNG
(CHEMBL2037349)
Show SMILES Clc1cccc(c1)-n1sc(=O)n(Cc2ccccc2)c1=O
Show InChI InChI=1S/C15H11ClN2O2S/c16-12-7-4-8-13(9-12)18-14(19)17(15(20)21-18)10-11-5-2-1-3-6-11/h1-9H,10H2
PDB
MMDB

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PC cid
PC sid
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n/an/a 1.09E+4n/an/an/an/an/an/a



TBA

Curated by ChEMBL


Assay Description
Inhibition of RGS8 interaction with Galpha0 protein by flow cytometry protein interaction assay


ACS Med Chem Lett 3: 146-150 (2012)


Article DOI: 10.1021/ml200263y
BindingDB Entry DOI: 10.7270/Q2NS0VXW
More data for this
Ligand-Target Pair
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